Activators

Ion Channels in Pain

Activators
Displaying 21 to 40 (out of 88 products)
  • ATX-II

    A Modulator of NaV Channels

    Cat # STA-700
    MW 4935 Da.
    Target Various NaV channels
  • BomoTx Toxin

    A Somatosensory, Pain Inducing Neuron Stimulator, Indirect P2X2/P2X3 Receptor Agonist

    Cat # NTB-200
    MW 13,834 Da.
    Target P2X2/P2X3 receptors
  • Cannabichromene

    An Activator of TRPA1 Channels and an Antagonist of Cannabinoid Receptor 1 and TRPM8 Channels

    Cat # C-315
    Source Synthetic
    MW 314.5
    Target TRPA1, TRPM8 channels, Cannabinoid receptor 1
  • Cannabidiol

    An Activator of TRPV1, TRPV3 and TRPA1 Channels and an Antagonist of Cannabinoid Receptors

    Cat # C-320
    Source Natural
    MW 314.46
    Target TRPV1, TRPV3, TRPA1 channels, CB receptors
  • Capsaicin

    A Powerful TRPV1 Agonist

    Cat # C-125
    Source Natural (from Capsicum sp.)
    MW 305.4
    Target TRPV1 channels
  • Capsiate

    A TRPA1 and TRPV1 Channel Activator

    Cat # C-255
    Source Natural
    MW 306.4
    Target TRPA1, TRPV1 channels
  • Celecoxib

    A Blocker of CaV1 Channels, a COX-2 Inhibitor and an Opener of KCNQ Channels 

    Cat # C-190
    Source Synthetic
    MW 381.4
    Target L-type Ca2+ and KCNQ channels
  • CGS 20625

    A Partial Agonist of GABA(A) Receptors

    Cat # C-390
    Source Synthetic
    MW 309.36
    Target GABA(A) receptors
  • Chlormethiazole hydrochloride

    A Positive Modulator of GABA(A) and Glycine Receptors

    Cat # C-360
    Source Synthetic
    MW 198.11
    Target GABA(A), Glycine receptors
  • Cono AIVGRPRF-amide

    A Specific Potentiator of ASIC3 Channel

    Cat # STC-174
    MW 914 Da.
    Target ASIC3 channel
  • Cono RPRF-amide

    A Specific Potentiator of ASIC3 Channel

    Cat # STC-170
    MW 574 Da.
    Target ASIC3 channel
  • Cono VGRPRF-amide

    A Specific Potentiator of ASIC3 Channel

    Cat # STC-172
    MW 730 Da.
    Target ASIC3 channel
  • Curcumin

    An Activator of TRPA1 Channels

    Cat # C-230
    Source Natural
    MW 368.4
    Target TRPA1 channels
  • (-)-Cytisine

    A nAChR Agonist and a Partial Agonist of β2 Subunit

    Cat # C-130
    Source Synthetic
    MW 190.2
    Target nAChR
  • Diazepam

    An Agonist of GABA(A) Receptors

    Cat # D-215
    Source Synthetic
    MW 284.74
    Target GABA(A) receptors
  • Diclofenac

    An Opener of KCNQ Channels

    Cat # D-180
    Source Synthetic
    MW 296.1
    Target KCNQ channels
  • DMAB-anabaseine dihydrochloride

    Antagonist or Partial Agonist of nAChR

    Cat # D-110
    Source Synthetic
    MW 364.3
    Target nAChR
  • Etodolac

    A Selective Activator of TRPA1 Channel

    Cat # E-140
    Source Synthetic
    MW 287.3
    Target TRPA1 channel
  • Flupirtine Maleate

    A Potent and Selective Modulator of KCNQ Channels

    Cat # F-150
    Source Synthetic
    MW 420.4
    Target KCNQ K+ channels
  • Ganaxolone

    A Selective Positive Modulator of GABA(A) Receptors

    Cat # G-120
    Source Synthetic
    MW 332.5
    Target GABA(A) receptors

* See product page

Displaying 21 to 40 (out of 88 products)