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Epilepsy

Blockers
Displaying 1 to 182 products (out of 182 products)

  • Slotoxin

    A Blocker of KCa1.1 Channel

    Cat # STS-410
    MW 4086 Da.
    Target KCa1.1 K+ channels
    More info
    • Bioassay Tested

  • 4-Aminopyridine

    A Non-Specific K+ Channel Blocker

    Cat # A-115
    Source Synthetic
    MW 94.1
    Target KV K+ channels
    More info
    • Bioassay Tested

  • 4,9-Anhydrotetrodotoxin

    A Potent and Selective Blocker of NaV1.6 Channel

    Cat # T-560
    Source Synthetic
    MW 301.25
    Target NaV1.6 channel
    More info
    • Bioassay Tested

  • 5,7-Dichlorokynurenic acid

    An Antagonist of NMDA Receptors

    Cat # D-190
    Source Synthetic
    MW 258.06
    Target NMDA receptors
    More info
    • Bioassay Tested

  • 5,7-Dichlorokynurenic acid monohydrate

    An Antagonist of NMDA Receptors

    Cat # D-191
    Source Synthetic
    MW 276.07
    Target NMDA receptors
    More info
    • Bioassay Tested

  • 7-Chlorokynurenic acid

    An Antagonist of NMDA Receptors

    Cat # C-285
    Source Synthetic
    MW 223.61
    Target NMDA receptors
    More info
    • Bioassay Tested

  • 7-Chlorokynurenic acid sodium salt

    An Antagonist of NMDA Receptors

    Cat # C-286
    Source Synthetic
    MW 245.59
    Target NMDA receptors
    More info
    • Bioassay Tested

  • α-Asarone

    An Antagonist of NaV Channels, GABA(A) Receptors, NMDA Receptors and an Inhibitor of TrkB Receptor

    Cat # A-260
    Source Natural
    MW 208.3
    Target NaV channels, GABA(A) receptors, TrkB receptors, NMDA receptors
    More info
    • Bioassay Tested

  • α-Bungarotoxin

    A Potent Antagonist of α7 and Muscle nAChR and GABA(A) Receptor Subtypes

    Cat # B-100
    MW 7984 Da.
    Target α7, α1/β1/γ/δ nAChR, GABA(A) receptor subtypes
    More info
    • Bioassay Tested

  • α-Bungarotoxin-ATTO Fluor-488

    A Fluorescent Conjugate for Sensitive Detection of Neuromuscular Junctions, GABA(A) Receptors, nAChRs, and α-Bungarotoxin Binding Sites

    Cat # B-100-AG
    MW ~9140 Da
    Target α7, α1/β1/γ/δ nAChR and GABA(A) receptor subtypes
    More info
    • Bioassay Tested

  • α-Bungarotoxin-ATTO Fluor-633

    A Fluorescent Conjugate for Sensitive Detection of Neuromuscular Junctions, GABA(A) Receptors, nAChRs, and α-Bungarotoxin Binding Sites

    Cat # B-100-FR
    MW ~9140 Da.
    Target α7, α1/β1/γ/δ nAChR and GABA(A) receptor subtypes
    More info
    • Bioassay Tested

  • α-Bungarotoxin-Biotin

    A Biotinylated Conjugate for Sensitive Detection of Neuromuscular Junctions, GABA(A) Receptors, nAChRs, and α-Bungarotoxin Binding Sites

    Cat # B-100-B
    MW ~9030 Da
    Target α7, α1/β1/γ/δ nAChR, GABA(A) receptor subtypes
    More info
    • Bioassay Tested

  • α-Bungarotoxin-FITC

    A Fluorescent Conjugate for Sensitive Detection of Neuromuscular Junctions, GABA(A) Receptors, nAChRs, and α-Bungarotoxin Binding Sites

    Cat # B-100-F
    MW ~8406 Da.
    Target α7, α1/β1/γ/δ nAChR and GABA(A) receptor subtypes
    More info
    • Bioassay Tested

  • α-Conotoxin ImI

    A Potent Antagonist of Mammalian α3/β2 Neuronal nAChR

    Cat # C-290
    MW 1351 Da.
    Target α3/β2 nAChR
    More info
    • Bioassay Tested

  • α-Conotoxin ImI-ATTO Fluor-590

    A Potent Antagonist of Mammalian α3/β2 nAChR Conjugated to the Fluorescent Dye ATTO-590

    Cat # C-290-AR
    MW 1924 Da.
    Target α3/β2 nAChR
    More info
    • Bioassay Tested

  • α-Conotoxin LtIA

    A Novel Antagonist of α3/β2 nAChR

    Cat # STC-550
    MW 1601.8 Da.
    Target α3/β2 nAChR
    More info
    • Bioassay Tested

  • α-Conotoxin PeIA

    An Antagonist of nAChR and N-Type Ca2+ Channels

    Cat # STC-970
    MW 1652 Da.
    Target nAChR, CaV2.2 Ca2+ channels
    More info
    • Bioassay Tested

  • κ-Conotoxin RIIIJ

    Voltage-Gated K+ Channel Blocker

    Cat # STC-660
    MW 2807.9 Da.
    Target KV1.2 K+ channels
    More info
    • Bioassay Tested

  • κ-Conotoxin RIIIK

    A Specific Potent Blocker of KV1.2 K+ Channels

    Cat # STC-650
    MW 2648 Da.
    Target KV1.2 K+ channels
    More info
    • Bioassay Tested

  • µ-Conotoxin BuIIIA

    A Selective and Potent Blocker of NaV1.2 and NaV1.4 Channels

    Cat # STC-540
    MW 2752 Da.
    Target NaV1.2, NaV1.4 channels
    More info
    • Bioassay Tested

  • µ-Conotoxin BuIIIB

    A Blocker of NaV1.4 and NaV1.3 and NaV1.2 Na+ Channels

    Cat # STC-661
    MW 2764 Da.
    Target NaV1.2, NaV1.3 and NaV1.4 Na+ channels
    More info
    • Bioassay Tested

  • µ-Conotoxin CnIIIC

    A Blocker of NaV Channels and an Antagonist of nAChRs

    Cat # STC-640
    MW 2376 Da.
    Target NaV Na+ channels, α3/β2 nAChR
    More info
    • Bioassay Tested

  • µ-Conotoxin KIIIA

    A Potent Blocker of Mammalian TTX-Sensitive NaV1 Channels

    Cat # C-280
    MW 1883 Da.
    Target TTX-sensitive Na+ channels
    More info
    • Bioassay Tested

  • µ-Conotoxin PIIIA

    A Potent Blocker of NaV1.2, NaV1.4 and NaV1.7 Na+ Channels

    Cat # STC-400
    MW 2604 Da.
    Target Various NaV channels
    More info
    • Bioassay Tested

  • µ-Conotoxin SIIIA

    A Blocker of TTX-Sensitive NaV1.2, NaV1.3 and NaV1.4 Voltage-Gated Na+ Channels

    Cat # STC-450
    MW 2207 Da.
    Target NaV1.2, NaV1.3, NaV1.4 Na+ channels
    More info
    • Bioassay Tested

  • ω-Agatoxin IVA

    A Blocker of P/Q-Type CaV Channels

    Cat # STA-500
    MW 5202 Da.
    Target P-type Ca2+ channels
    More info
    • Bioassay Tested

  • ω-Agatoxin TK

    A Blocker of P/Q-Type CaV Channels

    Cat # STA-530
    MW 5273 Da.
    Target P-type and Q-type Ca2+ channels
    More info
    • Bioassay Tested

  • ω-Conotoxin CVIB

    A Blocker of N-, P/Q-Type Ca2+ Channels

    Cat # STC-410
    MW 2710 Da.
    Target N-, P/Q-type Ca2+ channels
    More info
    • Bioassay Tested

  • ω-Conotoxin CVIC

    A Blocker of N-, P/Q-Type Ca2+ Channels

    Cat # STC-420
    MW 2783 Da.
    Target N-, P/Q-type channels
    More info
    • Bioassay Tested

  • ω-Conotoxin MVIIC

    A Blocker of Presynaptic CaV (N- and P/Q-Type) Channels

    Cat # C-150
    MW 2750 Da.
    Target N-type and P/Q-type Ca2+ channels
    More info
    • Bioassay Tested

  • ω-Conotoxin MVIID

    A Blocker of N- and P-Type CaV Channels 

    Cat # STC-751
    MW 2695 Da.
    Target N-, P-type Ca2+ channels
    More info
    • Bioassay Tested

  • ω-Grammotoxin SIA

    A Novel Blocker of CaV2.1 (P-type) and CaV2.2 (N-type) Channels

    Cat # G-450
    MW 4109.7 Da.
    Target P-type and N-type Ca2+ channels
    More info
    • Bioassay Tested

  • Amentoflavone

    A Negative Allosteric Modulator of GABA(A) Receptors

    Cat # A-165
    Source Natural
    MW 538.46
    Target GABA(A) receptors
    More info
    • Bioassay Tested

  • AmmTx3 Toxin

    A Blocker of A-Type K+ Channels

    Cat # STA-305
    MW 3822 Da.
    Target KV4 K+ channels
    More info
    • Bioassay Tested

  • Apamin

    A Blocker of Small Conductance Ca2+-Activated K+ Channels (SK Type)

    Cat # STA-200
    MW 2028 Da.
    Target KCa2 K+ channels
    More info
    • Bioassay Tested

  • Apamin-Biotin

    A Blocker of Small Conductance Ca2+-Activated K+ Channels (SK Type) Conjugated to Biotin

    Cat # STA-200-B
    MW 2367 Da.
    Target KCa2 K+ channels
    More info
    • Bioassay Tested

  • Arcaine sulfate

    An Antagonist of NMDA Receptors

    Cat # A-285
    Source Synthetic
    MW 270.31
    Target NMDA receptors
    More info
    • Bioassay Tested

  • BDS-I

    A Blocker of KV3 Channels and a Modulator of NaV Channels

    Cat # STB-400
    MW 4708 Da.
    Target KV3 K+ channels, NaV Na+ channels
    More info
    • Bioassay Tested

  • BDS-II

    A Blocker of KV3 Channels and a Modulator of NaV Channels

    Cat # B-450
    MW 4776 Da.
    Target KV3 K+ channels, NaV Na+ channels
    More info
    • Bioassay Tested

  • Benidipine hydrochloride

    A Dihydropyridine Blocker of Voltage-Gated Ca2+ Channels

    Cat # B-120
    Source Synthetic
    MW 542
    Target CaV1, CaV3 Ca2+ channels
    More info
    • Bioassay Tested

  • (+)-Bicuculline

    A Potent Antagonist of GABA(A) Receptors

    Cat # B-135
    Source Synthetic
    MW 367.4
    Target GABA(A) receptors
    More info
    • Bioassay Tested

  • (-)-Bicuculline methiodide

    An Antagonist of GABA(A) Receptors

    Cat # B-136
    Source Synthetic
    MW 509.27
    Target GABA(A) receptors
    More info
    • Bioassay Tested

  • (-)-Bicuculline methochloride

    An Antagonist of GABA(A) Receptors

    Cat # B-137
    Source Synthetic
    MW 417.84
    Target GABA(A) receptors
    More info
    • Bioassay Tested

  • Bilobalide

    An Antagonist of 5-HT3A and GABA(A) Receptors

    Cat # B-145
    Source Natural
    MW 326.3
    Target 5-HT3A, GABA(A) receptors
    More info
    • Bioassay Tested

  • Ceratotoxin-1

    A Blocker of NaV channels

    Cat # STC-680
    MW 4044 Da.
    Target NaV channels
    More info
    • Bioassay Tested

  • Ceratotoxin-2

    A Potent Blocker of Central Nervous System Voltage-Gated Na+ Channels

    Cat # STC-100
    MW 4093 Da.
    Target NaV channels
    More info
    • Bioassay Tested

  • CGP-37849

    A Potent and Selective Antagonist of NMDA Receptors

    Cat # C-325
    Source Synthetic
    MW 209.14
    Target NMDA receptors
    More info
    • Bioassay Tested

  • CGS 19755

    An NMDA Receptor Antagonist

    Cat # C-310
    Source Synthetic
    MW 223.16
    Target NMDA receptors
    More info
    • Bioassay Tested

  • Charybdotoxin

    A Blocker of KV1.2, KV1.3 and KCa1.1 K+ Channels

    Cat # STC-325
    MW 4296 Da.
    Target KCa1.1, KV1.2, KV1.3 K+ channels
    More info
    • Bioassay Tested

  • Chlorotoxin

    An Inhibitor of Chloride Channels

    Cat # RTC-450
    MW 3996 Da.
    Target Chloride channels
    More info
    • Bioassay Tested

  • Chlorotoxin

    An Inhibitor of Chloride Channels

    Cat # STC-460
    MW 3995 Da.
    Target Chloride channels
    More info
    • Bioassay Tested

  • Clobenpropit dihydrobromide

    A Potent and Selective Antagonist of Histamine H3 Receptors and an Antagonist of NMDA Receptors

    Cat # C-345
    Source Synthetic
    MW 470.65
    Target Histamine H3, Histamine H4, NMDA receptors
    More info
    • Bioassay Tested

  • CNS-1102

    A Potent NMDA Receptor Antagonist

    Cat # C-305
    Source Synthetic
    MW 339.86
    Target NMDA receptors
    More info
    • Bioassay Tested

  • Co 102862

    A Potent, State-Dependent Blocker of Neuronal NaV Channels

    Cat # C-160
    Source Synthetic
    MW 273.3
    Target NaV Na+ channels
    More info
    • Bioassay Tested

  • Conantokin G

    A Selective and Competitive Antagonist of GluN2B Receptor

    Cat # STC-666
    MW 2264.2 Da.
    Target GluN2B receptor
    More info
    • Bioassay Tested

  • Conantokin R

    An Antagonist of GluN2A and GluN2B Receptors

    Cat # STC-777
    Source Synthetic peptide
    MW 3098 Da.
    Target GluN2B receptor
    More info
    • Bioassay Tested

  • CP 465022 hydrochloride

    A Selective, Non-Competitive Antagonist of AMPA Receptors and a Modulator of NaV1.6 Channels

    Cat # C-335
    Source Synthetic
    MW 499.4
    Target AMPA receptors, NaV1.6 Na+ channels
    More info
    • Bioassay Tested

  • (±)-CPP

    An NMDA Receptor Antagonist

    Cat # C-175
    Source Synthetic
    MW 252.2
    Target NMDA receptors
    More info
    • Bioassay Tested

  • D-AP5

    A Competitive NMDA Receptor Antagonist

    Cat # D-145
    Source Synthetic
    MW 197.1
    Target NMDA receptors
    More info
    • Bioassay Tested

  • DL-AP5

    A Competitive NMDA Receptor Antagonist

    Cat # D-140
    Source Synthetic
    MW 197.1
    Target NMDA receptors
    More info
    • Bioassay Tested

  • DL-AP7

    An Antagonist of NMDA Receptors

    Cat # D-200
    Source Synthetic
    MW 225.19
    Target NMDA receptors
    More info
    • Bioassay Tested

  • α-Dendrotoxin

    A Blocker of KV1.1, KV1.2, KV1.6 and ASIC Channels

    Cat # D-350
    MW 7048 Da.
    Target KV1.1, KV1.2, KV1.6, ASIC channels
    More info
    • Bioassay Tested

  • β-Dendrotoxin

    A Potent Blocker of KV1.1 and KV1.2 Channels

    Cat # D-360
    MW ~7000 Da.
    Target KV1.1, KV1.2 K+ channels
    More info
    • Bioassay Tested

  • γ-Dendrotoxin

    A Potent Blocker of KV1.1 and KV1.2 Channels

    Cat # D-370
    MW ~7000 Da.
    Target KV1.1, KV1.2 K+ channels
    More info
    • Bioassay Tested

  • δ-Dendrotoxin

    A Potent and Specific Blocker of KV1.1 Channels and a Less Potent Blocker of Kir1.1 (ROMK1) Channels

    Cat # D-380
    MW 6568 Da.
    Target KV1.1, KV1.6 and Kir1.1 K+ channels
    More info
    • Bioassay Tested

  • Dendrotoxin-I

    A Potent Blocker of KV1.1 and KV1.2 Channels

    Cat # D-390
    MW 7149 Da.
    Target KV1.1, KV1.2 K+ channels
    More info
    • Bioassay Tested

  • Dendrotoxin-K

    A Potent Blocker of KV1.1 and KV1.2 Channels

    Cat # D-400
    MW 6560 Da.
    Target KV1.1, KV1.2 K+ channels
    More info
    • Bioassay Tested

  • Eliprodil

    An Antagonist of NMDA Receptors and N- and P-Type CaV Channels

    Cat # E-155
    Source Synthetic
    MW 347.9
    Target NMDA receptors, N-, P-type CaV channels
    More info
    • Bioassay Tested

  • Etbicyphat

    An Antagonist of GABA(A) Receptors

    Cat # E-175
    Source Synthetic
    MW 178.12
    Target GABA(A) receptors
    More info
    • Bioassay Tested

  • FTX-3.3

    A Blocker of P-Type CaV Channels

    Cat # F-120
    Source Synthetic
    MW 273.4
    Target P-type Ca2+ channels
    More info
    • Bioassay Tested

  • sFTX-3.3

    A Blocker of P-Type CaV Channels

    Cat # F-130
    Source Synthetic
    MW 287.4
    Target P-type Ca2+ channels
    More info
    • Bioassay Tested

  • GABA(A)-Compound 1b

    A Novel Antagonist of GABA(A) Receptors

    Cat # CMG-004
    Source Synthetic
    MW 415.39
    Target GABA(A) receptors
    More info
    • Bioassay Tested

  • Gabazine

    An Antagonist of GABA(A) and Glycine Receptors

    Cat # G-215
    Source Synthetic
    MW 287.32
    Target GABA(A), Glycine receptors
    More info
    • Bioassay Tested

  • Gabazine hydrobromide

    An Antagonist of GABA(A) and Glycine Receptors

    Cat # G-216
    Source Synthetic
    MW 368.23
    Target GABA(A), Glycine receptors
    More info
    • Bioassay Tested

  • GpTx-1

    A Blocker of NaV1.7, NaV1.5 and NaV1.4 Na+ Channels

    Cat # STG-400
    MW 4073.9 Da.
    Target NaV1.7, NaV1.5, NaV1.4 channels
    More info
    • Bioassay Tested

  • GrTx1

    A Blocker of NaV and KV11.1 Channels

    Cat # STG-250
    MW 3697 Da.
    Target NaV, KV11.1 channels
    More info
    • Bioassay Tested

  • GsAF-I

    A Blocker of TTX-Sensitive NaV and KV11.1 Channels

    Cat # STG-300
    MW 3707.9 Da.
    Target TTX-sensitive NaV, KV11.1 channels
    More info
    • Bioassay Tested

  • GsAF-II

    A Blocker of TTX-Sensitive NaV and KV11.1 Channels

    Cat # STG-350
    MW 3979.9 Da.
    Target TTX-sensitive NaV, KV11.1 channels
    More info
    • Bioassay Tested

  • GsMTx-4

    A Blocker of NaV1.7, TRPC1, TRPC6 and Piezo1 Channels

    Cat # STG-100
    MW 4096 Da.
    Target NaV1.7 channels, TRPC1, TRPC6, Piezo1
    More info
    • Bioassay Tested

  • GTx1-15

     A Blocker of Voltage-Gated Na+ and T-Type Ca2+ Channels

    Cat # STT-300
    MW 4075 Da.
    Target NaV Na+ Channels, T-type Ca2+ channels
    More info
    • Bioassay Tested

  • Guangxitoxin-1E

    A Potent Gating Modifier of KV2.1, KV2.2 and KV4.3 K+ Channels

    Cat # STG-200
    MW 3948.7 Da.
    Target Various KV channels
    More info
    • Bioassay Tested

  • Hainantoxin-III

    A Potent Mammalian TTX-Sensitive Voltage-Gated Na+ Channel Blocker

    Cat # STH-120
    MW 3608 Da.
    Target TTX-sensitive NaV Na+ channels
    More info
    • Bioassay Tested

  • Hainantoxin-IV

    A Blocker of TTX-Sensitive NaV Channels

    Cat # STH-130
    MW 3987 Da.
    Target TTX-sensitive NaV channels
    More info
    • Bioassay Tested

  • Haplotoxin-2

    A Blocker of NaV1.3 Na+ Channel and HERG K+ Channel

    Cat # STT-200
    MW 3708 Da.
    Target NaV1.3 Na+ channels, KV11.1 K+ channels
    More info
    • Bioassay Tested

  • Hd1a Toxin

    A Selective Blocker of NaV1.7 Channels

    Cat # STH-200
    MW 3822 Da.
    Target NaV1.7 channel
    More info
    • Bioassay Tested

  • Hemitoxin

    A Potent Blocker of KV1.1, KV1.2 and KV1.3 K+ Channels

    Cat # STH-500
    MW 3898 Da.
    Target KV1.1, KV1.2, KV1.3 K+ channels
    More info
    • Bioassay Tested

  • Heteropodatoxin-2

    A Potent Blocker of KV4 K+ Channels

    Cat # STH-340
    MW 3413 Da.
    Target KV4 K+ channels
    More info
    • Bioassay Tested

  • Hongotoxin-1

    A Potent Blocker of Some KV1 K+ Channels

    Cat # STH-400
    MW 4220 Da.
    Target KV1.1, KV1.2, KV1.3 K+ channels
    More info
    • Bioassay Tested

  • Huwentoxin-I

    An Antagonist of TTX-Sensitive NaV Channels, N-Type Ca2+ Channels and nAChRs

    Cat # STH-050
    MW 3750 Da.
    Target N-type CaV, TTX-sensitive NaV channels, nAChR
    More info
    • Bioassay Tested

  • Huwentoxin-IV

    A Potent Blocker of Neuronal TTX-Sensitive Voltage-Gated Na+ Channel

    Cat # STH-100
    MW 4106 Da.
    Target TTX-sensitive Na+ channels
    More info
    • Bioassay Tested

  • mHuwentoxin-IV

    A Blocker of TTX-Sensitive NaV Channels

    Cat # STH-101
    MW 4089 Da.
    Target TTX-sensitive Na+ channels
    More info
    • Bioassay Tested

  • m3-Huwentoxin IV

    A Potent and Selective NaV1.7 Channel Blocker

    Cat # STH-102
    MW 3988 Da.
    Target NaV1.7 channel
    More info
    • Bioassay Tested

  • Iberiotoxin

    A Potent and Specific Blocker of KCa1.1 K+ Channels

    Cat # STI-400
    MW 4230.9 Da.
    Target KCa1.1 K+ channels
    More info
    • Bioassay Tested

  • ICA 121431

    A Potent and Selective Blocker of NaV1.3 and NaV1.1 Channels

    Cat # I-170
    Source Synthetic
    MW 449.5
    Target NaV1.1, NaV1.3 channels
    More info
    • Bioassay Tested

  • Jingzhaotoxin-III

    A Blocker of KV2.1 and NaV1.5 Channels

    Cat # STJ-200
    MW 3919 Da.
    Target NaV1.5, KV2.1 channels
    More info
    • Bioassay Tested

  • Jingzhaotoxin-V

    A Potent Inhibitor of NaV Channels and KV4.2 and KV4.3 Channels

    Cat # STJ-050
    MW 3605.4 Da.
    Target NaV channels, KV4.2, KV4.3 channels
    More info
    • Bioassay Tested

  • Jingzhaotoxin-IX

    A Blocker of NaV1.4, NaV1.5 and KV2.1 Channels

    Cat # STJ-300
    MW 3953 Da.
    Target NaV1.4, NaV1.5, KV2.1 channels
    More info
    • Bioassay Tested

  • Jingzhaotoxin XI

    A Blocker of NaV1.5 and KV2.1 Channels

    Cat # STJ-400
    MW 3726 Da.
    Target KV2.1 and NaV1.5 channels
    More info
    • Bioassay Tested

  • Kaliotoxin-1

    A Powerful Blocker of KCa1.1 and certain KV1 Channels

    Cat # STK-370
    MW 4150 Da.
    Target KCa1.1 and some KV1 K+ channels
    More info
    • Bioassay Tested

  • KC 12291 hydrochloride

    An Orally Effective Cardioprotective NaV Channel Blocker

    Cat # K-105
    Source Synthetic
    MW 449.99
    Target NaV channels
    More info
    • Bioassay Tested

  • Kynurenic acid

    An Antagonist of Ionotropic Glutamate Receptors and α7 nAChR

    Cat # K-110
    Source Synthetic
    MW 189.2
    Target iGluR, α7 nAChR
    More info
    • Bioassay Tested

  • L-689,560

    A Potent and Selective Antagonist of NMDA Receptors

    Cat # L-225
    Source Synthetic
    MW 380.23
    Target NMDA receptors
    More info
    • Bioassay Tested

  • L-Ascorbic acid

    A Blocker of T-Type CaV Channels

    Cat # L-140
    Source Synthetic
    MW 176.1
    Target T-type Ca2+ channels
    More info
    • Bioassay Tested

  • Linopirdine

    A Blocker of KCNQ (KV7) Channels

    Cat # L-155
    Source Synthetic
    MW 391.46
    Target KCNQ K+ channels
    More info
    • Bioassay Tested

  • Linopirdine dihydrochloride

    A Blocker of KCNQ (KV7) Channels

    Cat # L-156
    Source Synthetic
    MW 464.39
    Target KCNQ K+ channels
    More info
    • Bioassay Tested

  • Maurotoxin

    A Potent Blocker of KCa and KV1 K+ Channels

    Cat # STM-340
    MW 3612 Da.
    Target KCa and KV1 K+ channels
    More info
    • Bioassay Tested

  • MCD peptide

    A Potent and Selective Blocker of KV1.1 and KV1.2 Channels

    Cat # STM-250
    MW 2588 Da.
    Target KV1.1, KV1.2 K+ channels
    More info
    • Bioassay Tested

  • Mibefradil dihydrochloride hydrate

    A Blocker of T-type CaV, Orai1-3, and KV10.1 Channels

    Cat # M-150
    Source Synthetic
    MW 568.55
    Target CaV3, Orai1-3, KV10.1 channels
    More info
    • Bioassay Tested

  • (+)-MK 801 maleate

    An Antagonist of NMDA Receptors

    Cat # M-230
    Source Synthetic
    MW 337.4
    Target NMDA receptors
    More info
    • Bioassay Tested

  • ML 218

    A Selective Blocker of T-type Channels

    Cat # M-165
    Source Synthetic
    MW 369.3
    Target T-type CaV channels
    More info
    • Bioassay Tested

  • ML 218 hydrochloride

    A Selective Blocker of T-type Channels

    Cat # M-166
    Source Synthetic
    MW 405.8
    Target T-type CaV channels
    More info
    • Bioassay Tested

  • MmTx1 Toxin

    A Super Potent Allosteric Modulator of GABA(A) Receptors

    Cat # STM-550
    MW 7205 Da.
    Target GABA(A) receptors
    More info
    • Bioassay Tested

  • MPX-004

    A Potent and Selective Antagonist of GluN2A-containing NMDA Receptors

    Cat # M-280
    Source Synthetic
    MW 455.91
    Target GluN2A-containing NMDA receptors
    More info
    • Bioassay Tested

  • N-Me-aminopyrimidinone 9

    A Specific Blocker of NaV1.7 Channel

    Cat # N-310
    Source Synthetic
    MW 303.4
    Target NaV1.7 channels
    More info
    • Bioassay Tested

  • NaV1.7-Compound 36

    A Potent and Selective Blocker of NaV1.7 Channels

    Cat # CMN-003
    Source Synthetic.
    MW 486.85
    Target NaV1.7 channels
    More info
    • Bioassay Tested

  • NNC 55-0396 dihydrochloride

    A Blocker of T-type CaV Channels

    Cat # N-205
    Source Synthetic
    MW 564.57
    Target T-type CaV channels
    More info
    • Bioassay Tested

  • NNC 55-0396 dihydrochloride hydrate

    A Blocker of T-type CaV Channels

    Cat # N-206
    Source Synthetic
    MW 573.48
    Target T-type CaV channels
    More info
    • Bioassay Tested

  • Noxiustoxin

    A Potent Blocker of KV1.2 and KV1.3 Channels

    Cat # STN-340
    MW 4194 Da.
    Target KV1.2, KV1.3 K+ channels
    More info
    • Bioassay Tested

  • NS8593

    A Blocker of KCa2 and TRPM7 Channels

    Cat # N-196
    Source Synthetic
    MW 263.3
    Target SK K+ channels, TRPM7
    More info
    • Bioassay Tested

  • NS8593 hydrochloride

    A Blocker of KCa2 and TRPM7 Channels

    Cat # N-195
    Source Synthetic
    MW 299.79
    Target SK K+ channels, TRPM7
    More info
    • Bioassay Tested

  • Oroxylin A

    An Antagonist of GABA(A) Receptors

    Cat # O-160
    Source Natural
    MW 284.26
    Target GABA(A) receptors
    More info
    • Bioassay Tested

  • OsK-1 Toxin

    A Potent Blocker of KV1.3 and KCa3.1 K+ Channels

    Cat # STO-150
    MW 4205 Da.
    Target KV1.1, KV1.2, KV1.3, and KCa3.1 K+ channels
    More info
    • Bioassay Tested

  • Pandinotoxin Kα

    A Blocker of A-Type and Shaker-Related Voltage-Gated K+ Channels

    Cat # STP-500
    MW 4033 Da.
    Target A-type and Shaker-related K+ channels
    More info
    • Bioassay Tested

  • Paxilline

    A Mycotoxin Blocker of KCa1.1 (BK) Channels and SERCA Pumps

    Cat # P-450
    Source Natural
    MW 435.6
    Target KCa K+ channels, SERCA pump
    More info
    • Bioassay Tested

  • PEAQX tetrasodium hydrate

    An Antagonist of NMDA Receptors

    Cat # P-255
    Source Synthetic
    MW 560.15
    Target NR1, NR2 receptors
    More info
    • Bioassay Tested

  • Penitrem A

    A Blocker of KCa1.1 (BK) Channels

    Cat # P-650
    Source Natural
    MW 634.2
    Target KCa1.1 K+ channels
    More info
    • Bioassay Tested

  • PF-04856264

    A Specific Blocker of NaV1.7 Channel

    Cat # P-265
    Source Synthetic
    MW 437.5
    Target NaV1.7 channels
    More info
    • Bioassay Tested

  • PF-05089771

    A Potent and Selective Blocker of NaV1.7 Channel

    Cat # P-315
    Source Synthetic
    MW 500.34
    Target NaV1.7 channels
    More info
    • Bioassay Tested

  • PF-05186462

    A Potent and Selective Blocker of NaV1.7 Channels

    Cat # P-365
    Source Synthetic
    MW 531.89
    Target NaV1.7 channels
    More info
    • Bioassay Tested

  • PF-05241328

    A Potent and Selective Blocker of NaV1.7 Channels

    Cat # P-345
    Source Synthetic
    MW 436.91
    Target NaV1.7 channels
    More info
    • Bioassay Tested

  • Phlo1a

    A Blocker of NaV1.7 Channels

    Cat # STP-350
    MW 4107 Da.
    Target NaV1.7 channels
    More info
    • Bioassay Tested

  • Phlo1b

    A Blocker of NaV1.7 Channels

    Cat # STP-370
    MW 4140 Da.
    Target NaV1.7 channels
    More info
    • Bioassay Tested

  • Phrixotoxin-1

    A Potent Blocker of KV4.2 and KV4.3 Channels

    Cat # STP-700
    MW 3549 Da.
    Target KV4.2, KV4.3 channels
    More info
    • Bioassay Tested

  • Phrixotoxin-2

    A Potent Blocker of KV4 Channels

    Cat # STP-710
    MW 3923 Da.
    Target KV4 channels
    More info
    • Bioassay Tested

  • Phrixotoxin-3

    A Potent Blocker of NaV1.2 and NaV1.6 Channels

    Cat # STP-720
    MW 4060 Da.
    Target NaV1.2, NaV1.6 channels
    More info
    • Bioassay Tested

  • Picrotoxin

    An Antagonist of GABA(A), Glycine, and 5-HT3 Receptors

    Cat # P-325
    Source Natural
    MW 602.58
    Target GABA(A), Glycine, 5-HT3 receptors
    More info
    • Bioassay Tested

  • Pilsicainide hydrochloride

    A Use-Dependent Anti-Arrhythmic NaV Channel Blocker

    Cat # P-145
    Source Synthetic
    MW 308.85
    Target TTX-Sensitive NaV channels
    More info
    • Bioassay Tested

  • ProTx-I

    A Blocker of NaV, CaV3.1, KV2.1 and TRPA1 Channels

    Cat # STP-400
    MW 3988 Da.
    Target NaV, CaV3.1, KV2.1, TRPA1 channels
    More info
    • Bioassay Tested

  • ProTx-II

    A Blocker of NaV1.7 and NaV1.5 Channels and Some T-Type Ca2+ Channels

    Cat # STP-100
    MW 3826.6 Da.
    Target NaV channels and T-type Ca2+ channels
    More info
    • Bioassay Tested

  • ProTx-II-Biotin

    A Blocker of NaV1.7 and NaV1.5 Channels and some T-Type Ca2+ Channels Conjugated to Biotin

    Cat # STP-100-B
    MW 4053 Da.
    Target NaV Na+ channels and T-type Ca2+ channels
    More info
    • Bioassay Tested

  • ProTx-III

    A Potent Blocker of NaV1.7 Channels

    Cat # STP-150
    MW 3802 Da
    Target NaV1.7 channels
    More info
    • Bioassay Tested

  • Pterinotoxin-1

    A Novel Blocker of NaV1.3, NaV1.7, and NaV1.8 Voltage-Gated Na+ Channels

    Cat # STT-100
    MW 3970 Da.
    Target NaV channels
    More info
    • Bioassay Tested

  • Pterinotoxin-2

    A Blocker of NaV1.3 and NaV1.7 Na+ Channels

    Cat # STT-150
    MW 3637 Da.
    Target NaV1.3, NaV1.7 Na+ channels
    More info
    • Bioassay Tested

  • Pyrrolopyrimidine 48

    A Blocker of NaV1.7 and NaV1.5 Channel

    Cat # P-275
    Source Synthetic
    MW 385.46
    Target NaV1.7, NaV1.5 channels
    More info
    • Bioassay Tested

  • QX-222 chloride

    A Blocker of NaV Channels

    Cat # Q-200
    Source Synthetic
    MW 256.77 (as net anhydrous)
    Target Various NaV Na+ channels
    More info
    • Bioassay Tested

  • QX-314 bromide

    A Local Anesthetic Blocker of Some NaV Channels

    Cat # Q-100
    Source Synthetic
    MW 343.3
    Target Various NaV  Na+ channels
    More info
    • Bioassay Tested

  • QX-314 chloride

    A Local Anesthetic Blocker of NaV Channels

    Cat # Q-150
    Source Synthetic
    MW 298.85
    Target Various NaV Na+ channels
    More info
    • Bioassay Tested

  • Ralfinamide mesylate

    A Use-Dependent Blocker of NaV Channels

    Cat # R-105
    Source Synthetic
    MW 398.5
    Target NaV Na+ channels
    More info
    • Bioassay Tested

  • Ro 8-4304 hydrochloride

    A Selective Antagonist of NMDA Receptors

    Cat # R-165
    Source Synthetic
    MW 406.88
    Target NMDA receptors
    More info
    • Bioassay Tested

  • Ro 25-6981 maleate

    A Potent and Selective Antagonist of GluN2B-Containing NMDA Receptors

    Cat # R-180
    Source Synthetic
    MW 455.55
    Target GluN2B
    More info
    • Bioassay Tested

  • Roscovitine

    A Cyclin-Dependent Kinase (CDK) Inhibitor and a T-Type CaV Channel Blocker

    Cat # R-300
    Source Synthetic
    MW 354.46
    Target CDKs, T-type CaV channels
    More info
    • Bioassay Tested

  • RY796

    A Blocker of KV2 Channels

    Cat # R-160
    Source Synthetic
    MW 353.5
    Target KV2 channels
    More info
    • Bioassay Tested

  • Scyllatoxin

    A Potent Blocker of KCa2 (SK) K+ Channels

    Cat # STS-370
    MW 3423 Da.
    Target KCa2 K+ channels
    More info
    • Bioassay Tested

  • SKF 96365 hydrochloride

    A Blocker of CaV3 and TRPC channels and STIM1

    Cat # S-175
    Source Synthetic
    MW 402.9
    Target CaV3 channels, TRPC, STIM1
    More info
    • Bioassay Tested

  • SNX-482

    A Blocker of CaV2.3 and KV4.3 Channels

    Cat # RTS-500
    MW 4495 Da.
    Target CaV2.3, CaV2.1, KV4.2, KV4.3 channels
    More info
    • Bioassay Tested

  • Spinoxin

    A Potent Blocker of KV1.2 and KV1.3 Channels

    Cat # STS-500
    MW 3701.2 Da.
    Target KV1.2, KV1.3 channels
    More info
    • Bioassay Tested

  • SsTx Toxin

    A Blocker of KCNQ and KV1.3 Channels

    Cat # STS-700
    MW 6018 Da.
    Target KCNQ1, KCNQ2, KCNQ4, KCNQ5, KV1.3 channels
    More info
    • Bioassay Tested

  • ShK (Stichodactyla Toxin)

    A Blocker of KV Channels

    Cat # STS-400
    MW 4055 Da.
    Target Various KV K+ channels
    More info
    • Bioassay Tested

  • Stichodactyla Toxin-ATTO Fluor-590

    Fluorescent ShK Conjugate for Sensitive Detection of KV Channels

    Cat # STS-400-AR
    MW ~ 4627 Da.
    Target KV1.1, KV1.3, KV1.4, KV1.6 channels
    More info
    • Bioassay Tested

  • Stichodactyla Toxin-Biotin

    Biotinylated ShK Conjugate for Sensitive Detection of KV Channels

    Cat # STS-400-B
    MW 4563 Da.
    Target KV1.1, KV1.3, KV1.4, KV1.6 channels
    More info
    • Bioassay Tested

  • Stromatoxin-1

    A Potent Blocker of KV2.1, KV2.2, KV4.2 and KV9.3 Channels

    Cat # STS-350
    MW 3792 Da.
    Target Various KV channels
    More info
    • Bioassay Tested

  • Tamapin

    A Blocker of KCa2 Channels

    Cat # STT-400
    MW 3458.16 Da.
    Target KCa2 K+ channels
    More info
    • Bioassay Tested

  • TCN 201

    An Antagonist of NMDA Receptors

    Cat # T-190
    Source Synthetic
    MW 461.89
    Target NMDA receptors
    More info
    • Bioassay Tested

  • TCN 213

    An Antagonist of NMDA Receptors

    Cat # T-215
    Source Synthetic
    MW 376.54
    Target NMDA receptors
    More info
    • Bioassay Tested

  • Tetrodotoxin citrate

    A Classic Blocker of a Subset of NaV Channels

    Cat # T-550
    Source Natural
    MW 319.27
    Target Various NaV channels
    More info
    • Bioassay Tested

  • Tetrodotoxin citrate free

    A Classic Blocker of a Subset of NaV Channels

    Cat # T-500
    Source Natural
    MW 319.28
    Target Various NaV Na+ channels
    More info
    • Bioassay Tested

  • Tityustoxin-Kα

    A KV1.2 Channel Blocker

    Cat # STT-360
    MW 3942 Da.
    Target KV1.2 K+ channels
    More info
    • Bioassay Tested

  • Tityustoxin-Kα-ATTO Fluor-594

    A KV1.2 K+ Channel Blocker Conjugated to the Fluorescent Dye ATTO-594

    Cat # STT-360-AR
    MW ~4900 Da.
    Target KV1.2 K+ channels
    More info
    • Bioassay Tested

  • Tracazolate hydrochloride

    A Modulator of GABA(A) Receptors

    Cat # T-230
    Source Synthetic
    MW 340.85
    Target GABA(A) receptors
    More info
    • Bioassay Tested

  • TTA-A2

    A Blocker of T-Type CaV Channels

    Cat # T-140
    Source Synthetic
    MW 378.39
    Target T-type CaV channels
    More info
    • Bioassay Tested

  • TTA-P2

    A Blocker of T-Type CaV Channels

    Cat # T-155
    Source Synthetic
    MW 431
    Target T-type CaV channels
    More info
    • Bioassay Tested

  • TTA-P2 (S-enantiomer)

    A Blocker of T-Type CaV Channels

    Cat # T-210
    Source Synthetic
    MW 431
    Target CaV3 channels
    More info
    • Bioassay Tested

  • U 93631

    An Antagonist of GABA(A) and 5-HT3A Receptors

    Cat # U-120
    Source Synthetic
    MW 299.37
    Target GABA(A), 5-HT3A receptors
    More info
    • Bioassay Tested

  • Urotoxin

    A Super Potent Blocker of KV1.2 Channel

    Cat # STU-200
    MW 4012.7 Da.
    Target KV1.2, KV1.1, KV1.3, KCa3.1 channels
    More info
    • Bioassay Tested

  • Verruculogen

    A Blocker of KCa1.1 (BK) Channels

    Cat # V-500
    Source Natural
    MW 511.23
    Target KCa1.1 K+ channels
    More info
    • Bioassay Tested

  • VSTX3

    A Blocker of NaV1.3, NaV1.7, NaV1.8 Voltage-Gated Na+ Channels

    Cat # STT-350
    MW 4172 Da.
    Target NaV1.3, NaV1.7, NaV1.8 Na+ channels
    More info
    • Bioassay Tested

  • Waglerin-1

    A Potent Antagonist of nAChR and a Modulator of GABA(A) Receptors

    Cat # STW-001
    MW 2520 Da.
    Target nAChR, GABA(A) receptors
    More info
    • Bioassay Tested

  • XE991

    A Blocker of KCNQ Channels

    Cat # X-100
    Source Synthetic
    MW 376.45
    Target KCNQ K+ channels
    More info
    • Bioassay Tested

  • XE991 dihydrochloride

    A Blocker of KCNQ Channels

    Cat # X-101
    Source Synthetic
    MW 449.37
    Target KCNQ K+ channels
    More info
    • Bioassay Tested

  • XEN907

    A Specific Blocker of NaV1.7 Channels

    Cat # X-105
    Source Synthetic
    MW 351.1
    Target NaV1.7 channels
    More info
    • Bioassay Tested

  • ZD 9379

    An Antagonist of NMDA Receptors

    Cat # Z-120
    Source Synthetic
    MW 383.79
    Target NMDA receptors
    More info
    • Bioassay Tested

  • GABA(A) Receptor Antagonist Explorer Kit

    A Screening Package of GABA(A) Receptor Antagonists Economically Priced

    Cat # EK-420
    More info

* See product page

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