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Ion Channels in Pain

Blockers
Displaying 1 to 188 products (out of 188 products)
  • Huwentoxin-XVI

    A Potent and Reversible Blocker of CaV2.2 Channels

    Cat # STH-105
    MW 4437 Da.
    Target N-type Ca2+ channels
    • Bioassay Tested
  • 4-Aminopyridine

    A Non-Specific K+ Channel Blocker

    Cat # A-115
    Source Synthetic
    MW 94.1
    Target KV K+ channels
    • Bioassay Tested
  • 4,9-Anhydrotetrodotoxin

    A Potent and Selective Blocker of NaV1.6 Channel

    Cat # T-560
    Source Synthetic
    MW 301.25
    Target NaV1.6 channel
    • Bioassay Tested
  • 5′-Iodoresiniferatoxin

    A Potent and Partial Blocker of TRPV1 Channel

    Cat # I-800
    Source Semi-synthetic
    MW 754.6
    Target TRPV1 channels
    • Bioassay Tested
  • α-Asarone

    An Antagonist of NaV Channels, GABA(A) Receptors, NMDA Receptors and an Inhibitor of TrkB Receptor

    Cat # A-260
    Source Natural
    MW 208.3
    Target NaV channels, GABA(A) receptors, TrkB receptors, NMDA receptors
    • Bioassay Tested
  • α-Bungarotoxin

    A Potent Antagonist of α7 and Muscle nAChR and GABA(A) Receptor Subtypes

    Cat # B-100
    MW 7984 Da.
    Target α7, α1/β1/γ/δ nAChR, GABA(A) receptor subtypes
    • Bioassay Tested
  • α-Bungarotoxin-ATTO Fluor-488

    A Fluorescent Conjugate for Sensitive Detection of Neuromuscular Junctions, GABA(A) Receptors, nAChRs, and α-Bungarotoxin Binding Sites

    Cat # B-100-AG
    MW ~9140 Da
    Target α7, α1/β1/γ/δ nAChR and GABA(A) receptor subtypes
    • Bioassay Tested
  • α-Bungarotoxin-ATTO Fluor-633

    A Fluorescent Conjugate for Sensitive Detection of Neuromuscular Junctions, GABA(A) Receptors, nAChRs, and α-Bungarotoxin Binding Sites

    Cat # B-100-FR
    MW ~9140 Da.
    Target α7, α1/β1/γ/δ nAChR and GABA(A) receptor subtypes
    • Bioassay Tested
  • α-Bungarotoxin-Biotin

    A Biotinylated Conjugate for Sensitive Detection of Neuromuscular Junctions, GABA(A) Receptors, nAChRs, and α-Bungarotoxin Binding Sites

    Cat # B-100-B
    MW ~9030 Da
    Target α7, α1/β1/γ/δ nAChR, GABA(A) receptor subtypes
    • Bioassay Tested
  • α-Bungarotoxin-FITC

    A Fluorescent Conjugate for Sensitive Detection of Neuromuscular Junctions, GABA(A) Receptors, nAChRs, and α-Bungarotoxin Binding Sites

    Cat # B-100-F
    MW ~8406 Da.
    Target α7, α1/β1/γ/δ nAChR and GABA(A) receptor subtypes
    • Bioassay Tested
  • α-Conotoxin AuIA

    An Antagonist of α3/β4 nAChR

    Cat # STC-960
    MW 1726 Da.
    Target α3/β4 nAChR
    • Bioassay Tested
  • α-Conotoxin AuIB

    A Potent Antagonist of Mammalian α3/β4 Neuronal nAChR

    Cat # STC-310
    MW 1572 Da.
    Target α3/β4 nAChR
    • Bioassay Tested
  • α-Conotoxin PeIA

    An Antagonist of nAChR and N-Type Ca2+ Channels

    Cat # STC-970
    MW 1652 Da.
    Target nAChR, CaV2.2 Ca2+ channels
    • Bioassay Tested
  • α-Conotoxin PIA

    A Selective nAChRα6 Antagonist

    Cat # STC-870
    MW 1981 Da
    Target α6 nAChR
    • Bioassay Tested
  • µ-Conotoxin BuIIIB

    A Blocker of NaV1.4 and NaV1.3 and NaV1.2 Na+ Channels

    Cat # STC-661
    MW 2764 Da.
    Target NaV1.2, NaV1.3 and NaV1.4 Na+ channels
    • Bioassay Tested
  • µ-Conotoxin CnIIIC

    A Blocker of NaV Channels and an Antagonist of nAChRs

    Cat # STC-640
    MW 2376 Da.
    Target NaV Na+ channels, α3/β2 nAChR
    • Bioassay Tested
  • µ-Conotoxin KIIIA

    A Potent Blocker of Mammalian TTX-Sensitive NaV1 Channels

    Cat # C-280
    MW 1883 Da.
    Target TTX-sensitive Na+ channels
    • Bioassay Tested
  • µ-Conotoxin PIIIA

    A Potent Blocker of NaV1.2, NaV1.4 and NaV1.7 Na+ Channels

    Cat # STC-400
    MW 2604 Da.
    Target Various Nachannels
    • Bioassay Tested
  • µ-Conotoxin SIIIA

    A Blocker of TTX-Sensitive NaV1.2, NaV1.3 and NaV1.4 Voltage-Gated Na+ Channels

    Cat # STC-450
    MW 2207 Da.
    Target NaV1.2, NaV1.3, NaV1.4 Na+ channels
    • Bioassay Tested
  • ω-Agatoxin IVA

    A Blocker of P/Q-Type CaV Channels

    Cat # STA-500
    MW 5202 Da.
    Target P-type Ca2+ channels
    • Bioassay Tested
  • ω-Agatoxin TK

    A Blocker of P/Q-Type CaV Channels

    Cat # STA-530
    MW 5273 Da.
    Target P-type and Q-type Ca2+ channels
    • Bioassay Tested
  • ω-Conotoxin CnVIIA

    A Specific Blocker of N-Type Ca2+ Channels 

    Cat # STC-800
    MW 2848 Da.
    Target N-type Ca2+ channels
    • Bioassay Tested
  • ω-Conotoxin CVIA

    A Blocker of N-Type CaV Channels 

    Cat # STC-750
    MW 2642 Da.
    Target CaV2.2 channels
    • Bioassay Tested
  • ω-Conotoxin CVIB

    A Blocker of N-, P/Q-Type Ca2+ Channels

    Cat # STC-410
    MW 2710 Da.
    Target N-, P/Q-type Ca2+ channels
    • Bioassay Tested
  • ω-Conotoxin CVIC

    A Blocker of N-, P/Q-Type Ca2+ Channels

    Cat # STC-420
    MW 2783 Da.
    Target N-, P/Q-type channels
    • Bioassay Tested
  • ω-Conotoxin CVIE

    A Blocker of N-Type Ca2+ Channels

    Cat # STC-760
    MW 2640 Da.
    Target N-Type Ca2+ channels
    • Bioassay Tested
  • ω-Conotoxin CVIF

    A Blocker of N-Type CaV Channels 

    Cat # STC-770
    MW 2665 Da.
    Target CaV2.2 channels
    • Bioassay Tested
  • ω-Conotoxin FVIA

    A Potent Blocker of CaV2.2 Channel

    Cat # STC-780
    MW 2567 Da.
    Target CaV2.2 channels
    • Bioassay Tested
  • ω-Conotoxin GVIA

    A Blocker of N-Type Ca2+ Channels

    Cat # C-300
    MW 3037 Da.
    Target N-type Ca2+ channels
    • Bioassay Tested
  • ω-Conotoxin MVIIA

    A Specific Blocker of CaV2.2 Channel

    Cat # C-670
    MW 2639.20 Da.
    Target CaV2.2 Ca2+ channel
    • Bioassay Tested
  • ω-Conotoxin MVIIC

    A Blocker of Presynaptic CaV (N- and P/Q-Type) Channels

    Cat # C-150
    MW 2750 Da.
    Target N-type and P/Q-type Ca2+ channels
    • Bioassay Tested
  • ω-Conotoxin MVIID

    A Blocker of N- and P-Type CaV Channels 

    Cat # STC-751
    MW 2695 Da.
    Target N-, P-type Ca2+ channels
    • Bioassay Tested
  • ω-Conotoxin RVIA

    A Blocker of CaV2.2 Ca2+ Channel

    Cat # STC-850
    MW 2915 Da.
    Target CaV2.2 Ca2+ channels
    • Bioassay Tested
  • ω-Conotoxin SO3

    A Blocker of N-Type Ca2+ Channels

    Cat # STC-470
    MW 2562 Da.
    Target CaV2.2 Ca2+ channels
    • Bioassay Tested
  • ω-Conotoxin SVIB

    A Potent Blocker of N-Type CaV Channels

    Cat # STC-160
    MW 2739 Da.
    Target N-Type CaV channels
    • Bioassay Tested
  • ω-Grammotoxin SIA

    A Novel Blocker of CaV2.1 (P-type) and CaV2.2 (N-type) Channels

    Cat # G-450
    MW 4109.7 Da.
    Target P-type and N-type Ca2+ channels
    • Bioassay Tested
  • A-317491 sodium salt hydrate

    A Selective Antagonist of P2X3 and P2X2/3 Receptors

    Cat # A-380
    Source Synthetic
    MW 565.57 (free acid, anhydrous)
    Target P2X3 receptors
    • Bioassay Tested
  • A 784168

    A Potent Blocker of TRPV1 Channel

    Cat # A-345
    Source Synthetic
    MW 479.4
    Target TRPV1 channel
    • Bioassay Tested
  • A-803467

    A Potent and Selective Blocker of the TTX-Resistant NaV1.8 Channel

    Cat # A-105
    Source Synthetic
    MW 357.8
    Target NaV1.8 Na+ channels
    • Bioassay Tested
  • A-889425

    A Blocker of TRPV1 Channels

    Cat # A-195
    Source Synthetic
    MW 425.4
    Target TRPV1 channels
    • Bioassay Tested
  • A 967079

    A Blocker of TRPA1 Channels

    Cat # A-225
    Source Synthetic
    MW 207.2
    Target TRPA1 channels
    • Bioassay Tested
  • AF-353

    A Potent and Selective Antagonist of P2X3 Receptor

    Cat # A-375
    Source Synthetic
    MW 400.21
    Target P2X3 receptors
    • Bioassay Tested
  • Amentoflavone

    A Negative Allosteric Modulator of GABA(A) Receptors

    Cat # A-165
    Source Natural
    MW 538.46
    Target GABA(A) receptors
    • Bioassay Tested
  • AMG-9090

    A Blocker of TRPA1, TRPV1 and TRPM8 Channels

    Cat # A-300
    Source Synthetic
    MW 395.12
    Target TRPA1, TRPM8, TRPV1 channels
    • Bioassay Tested
  • AmmTx3 Toxin

    A Blocker of A-Type K+ Channels

    Cat # STA-305
    MW 3822 Da.
    Target KV4 K+ channels
    • Bioassay Tested
  • AP-18

    A Reversible TRPA1 Channel Blocker

    Cat # A-250
    Source Synthetic
    MW 209.7
    Target TRPA1 channels
    • Bioassay Tested
  • Apamin

    A Blocker of Small Conductance Ca2+-Activated K+ Channels (SK Type)

    Cat # STA-200
    MW 2028 Da.
    Target KCa2 K+ channels
    • Bioassay Tested
  • Apamin-Biotin

    A Blocker of Small Conductance Ca2+-Activated K+ Channels (SK Type) Conjugated to Biotin

    Cat # STA-200-B
    MW 2367 Da.
    Target KCa2 K+ channels
    • Bioassay Tested
  • APETx2

    A Blocker of ASIC3 Channel

    Cat # STA-160
    MW 4561 Da.
    Target ASIC3 channels
    • Bioassay Tested
  • Arcaine sulfate

    An Antagonist of NMDA Receptors

    Cat # A-285
    Source Synthetic
    MW 270.31
    Target NMDA receptors
    • Bioassay Tested
  • (S)-ATPO

    An Antagonist of AMPA/Kainate Receptors

    Cat # A-330
    Source Synthetic
    MW 322.25
    Target AMPA/Kainate receptors
    • Bioassay Tested
  • BCTC

    A Potent Antagonist of TRPV1 and TRPM8 Channels

    Cat # B-110
    Source Synthetic
    MW 372.9
    Target TRPV1 and TRPM8 channels
    • Bioassay Tested
  • BDS-I

    A Blocker of KV3 Channels and a Modulator of NaV Channels

    Cat # STB-400
    MW 4708 Da.
    Target KV3 K+ channels, NaV Na+ channels
    • Bioassay Tested
  • Benidipine hydrochloride

    A Dihydropyridine Blocker of Voltage-Gated Ca2+ Channels

    Cat # B-120
    Source Synthetic
    MW 542
    Target CaV1, CaV3 Ca2+ channels
    • Bioassay Tested
  • (+)-Bicuculline

    A Potent Antagonist of GABA(A) Receptors

    Cat # B-135
    Source Synthetic
    MW 367.4
    Target GABA(A) receptors
    • Bioassay Tested
  • (-)-Bicuculline methiodide

    An Antagonist of GABA(A) Receptors

    Cat # B-136
    Source Synthetic
    MW 509.27
    Target GABA(A) receptors
    • Bioassay Tested
  • (-)-Bicuculline methochloride

    An Antagonist of GABA(A) Receptors

    Cat # B-137
    Source Synthetic
    MW 417.84
    Target GABA(A) receptors
    • Bioassay Tested
  • Bilobalide

    An Antagonist of 5-HT3A and GABA(A) Receptors

    Cat # B-145
    Source Natural
    MW 326.3
    Target 5-HT3A, GABA(A) receptors
    • Bioassay Tested
  • Cannabichromene

    An Activator of TRPA1 Channels and an Antagonist of Cannabinoid Receptor 1 and TRPM8 Channels

    Cat # C-315
    Source Synthetic
    MW 314.5
    Target TRPA1, TRPM8 channels, Cannabinoid receptor 1
    • Bioassay Tested
  • Capsazepine

    A Selective TRPV1 Blocker and an Activator of ENaCγ Channels

    Cat # C-120
    Source Synthetic
    MW 376.9
    Target TRPV1, ENaCγ channels
    • Bioassay Tested
  • Ceratotoxin-1

    A Blocker of NaV channels

    Cat # STC-680
    MW 4044 Da.
    Target NaV channels
    • Bioassay Tested
  • Ceratotoxin-2

    A Potent Blocker of Central Nervous System Voltage-Gated Na+ Channels

    Cat # STC-100
    MW 4093 Da.
    Target NaV channels
    • Bioassay Tested
  • Chelerythrine chloride

    An Inhibitor of Protein Kinase C, SERCA Pump, and P2X7 Receptor

    Cat # C-400
    Source Natural
    MW 383.84
    Target PKC, SERCA pumps, P2X7 receptor
    • Bioassay Tested
  • Chembridge-5861528

    A Selective Blocker of TRPA1 Channel

    Cat # C-235
    Source Synthetic
    MW 369.4
    Target TRPA1 channels
    • Bioassay Tested
  • Cilnidipine

    A Blocker of L- and N-Type CaV Channels 

    Cat # C-135
    Source Synthetic
    MW 492.5
    Target L- and N-type Ca2+ channels
    • Bioassay Tested
  • CNQX

    AMPA/Kainate Receptor Antagonist

    Cat # C-140
    Source Synthetic
    MW 232.2
    Target AMPA/Kainate receptors
    • Bioassay Tested
  • CNQX disodium salt

    AMPA/Kainate Receptor Antagonist

    Cat # C-141
    Source Synthetic
    MW 276.1
    Target AMPA/Kainate receptors
    • Bioassay Tested
  • CNS-1102

    A Potent NMDA Receptor Antagonist

    Cat # C-305
    Source Synthetic
    MW 339.86
    Target NMDA receptors
    • Bioassay Tested
  • Co 102862

    A Potent, State-Dependent Blocker of Neuronal NaV Channels

    Cat # C-160
    Source Synthetic
    MW 273.3
    Target NaV Na+ channels
    • Bioassay Tested
  • Conantokin G

    A Selective and Competitive Antagonist of GluN2B Receptor

    Cat # STC-666
    MW 2264.2 Da.
    Target GluN2B receptor
    • Bioassay Tested
  • Conantokin R

    An Antagonist of GluN2A and GluN2B Receptors

    Cat # STC-777
    Source Synthetic peptide
    MW 3098 Da.
    Target GluN2B receptor
    • Bioassay Tested
  • (±)-CPP

    An NMDA Receptor Antagonist

    Cat # C-175
    Source Synthetic
    MW 252.2
    Target NMDA receptors
    • Bioassay Tested
  • α-Dendrotoxin

    A Blocker of KV1.1, KV1.2, KV1.6 and ASIC Channels

    Cat # D-350
    MW 7048 Da.
    Target KV1.1, KV1.2, KV1.6, ASIC channels
    • Bioassay Tested
  • β-Dendrotoxin

    A Potent Blocker of KV1.1 and KV1.2 Channels

    Cat # D-360
    MW ~7000 Da.
    Target KV1.1, KV1.2 K+ channels
    • Bioassay Tested
  • γ-Dendrotoxin

    A Potent Blocker of KV1.1 and KV1.2 Channels

    Cat # D-370
    MW ~7000 Da.
    Target KV1.1, KV1.2 K+ channels
    • Bioassay Tested
  • δ-Dendrotoxin

    A Potent and Specific Blocker of KV1.1 Channels and a Less Potent Blocker of Kir1.1 (ROMK1) Channels

    Cat # D-380
    MW 6568 Da.
    Target KV1.1, KV1.6 and Kir1.1 K+ channels
    • Bioassay Tested
  • Dendrotoxin-I

    A Potent Blocker of KV1.1 and KV1.2 Channels

    Cat # D-390
    MW 7149 Da.
    Target KV1.1, KV1.2 K+ channels
    • Bioassay Tested
  • Dendrotoxin-K

    A Potent Blocker of KV1.1 and KV1.2 Channels

    Cat # D-400
    MW 6560 Da.
    Target KV1.1, KV1.2 K+ channels
    • Bioassay Tested
  • D-AP5

    A Competitive NMDA Receptor Antagonist

    Cat # D-145
    Source Synthetic
    MW 197.1
    Target NMDA receptors
    • Bioassay Tested
  • DL-AP5

    A Competitive NMDA Receptor Antagonist

    Cat # D-140
    Source Synthetic
    MW 197.1
    Target NMDA receptors
    • Bioassay Tested
  • 5-(N,N-Dimethyl)amiloride hydrochloride

    A Blocker of TRPA1 Channels and Selective Blocker of Na+/H+ and Na+/Ca2+ Exchangers

    Cat # D-165
    Source Synthetic
    MW 294.1
    Target TRPA1 channel, Na+/H+ and Na+/Ca2+ exchangers
    • Bioassay Tested
  • DNQX

    AMPA/Kainate Receptor Antagonist

    Cat # D-131
    Source Synthetic
    MW 252.1
    Target AMPA/kainate receptors
    • Bioassay Tested
  • DNQX disodium salt

    AMPA/Kainate Receptor Antagonist

    Cat # D-130
    Source Synthetic
    MW 296.1
    Target AMPA/kainate receptors
    • Bioassay Tested
  • Evans Blue tetrasodium salt

    An Antagonist of AMPA/Kainate receptors, P2X Receptors and a Potent Inhibitor of L-Glutamate Uptake

    Cat # E-110
    Source Synthetic
    MW 960.8
    Target AMPA, Kainate, P2X receptors
    • Bioassay Tested
  • FTX-3.3

    A Blocker of P-Type CaV Channels

    Cat # F-120
    Source Synthetic
    MW 273.4
    Target P-type Ca2+ channels
    • Bioassay Tested
  • GpTx-1

    A Blocker of NaV1.7, NaV1.5 and NaV1.4 Na+ Channels

    Cat # STG-400
    MW 4073.9 Da.
    Target NaV1.7, NaV1.5, NaV1.4 channels
    • Bioassay Tested
  • GsMTx-4

    A Blocker of NaV1.7, TRPC1, TRPC6 and Piezo1 Channels

    Cat # STG-100
    MW 4096 Da.
    Target NaV1.7 channels, TRPC1, TRPC6, Piezo1
    • Bioassay Tested
  • GTx1-15

     A Blocker of Voltage-Gated Na+ and T-Type Ca2+ Channels

    Cat # STT-300
    MW 4075 Da.
    Target NaV Na+ Channels, T-type Ca2+ channels
    • Bioassay Tested
  • GYKI 52466 hydrochloride

    An Antagonist of AMPA and Kainate Receptors

    Cat # G-125
    Source Synthetic
    MW 329.78
    Target AMPA/Kainate receptors
    • Bioassay Tested
  • GYKI 53655 hydrochloride

    An Antagonist of AMPA and Kainate Receptors

    Cat # G-220
    Source Synthetic
    MW 388.85
    Target AMPA, Kainate receptors
    • Bioassay Tested
  • Hainantoxin-III

    A Potent Mammalian TTX-Sensitive Voltage-Gated Na+ Channel Blocker

    Cat # STH-120
    MW 3608 Da.
    Target TTX-sensitive NaV Na+ channels
    • Bioassay Tested
  • Hainantoxin-IV

    A Blocker of TTX-Sensitive NaV Channels

    Cat # STH-130
    MW 3987 Da.
    Target TTX-sensitive NaV channels
    • Bioassay Tested
  • HC-030031

    A Selective TRPA1 Channel Blocker

    Cat # H-105
    Source Synthetic
    MW 355.4
    Target TRPA1 channels
    • Bioassay Tested
  • Hemitoxin

    A Potent Blocker of KV1.1, KV1.2 and KV1.3 K+ Channels

    Cat # STH-500
    MW 3898 Da.
    Target KV1.1, KV1.2, KV1.3 K+ channels
    • Bioassay Tested
  • Heteropodatoxin-2

    A Potent Blocker of KV4 K+ Channels

    Cat # STH-340
    MW 3413 Da.
    Target KV4 K+ channels
    • Bioassay Tested
  • Hm3a Toxin

    A Highly Potent ASIC1a Blocker and ASIC1b Activator

    Cat # STH-250
    MW 4287.1 Da.
    Target ASIC1a and ASIC1b
    • Bioassay Tested
  • HMA

    An Antagonist of Na+/H+ Exchangers, P2X7 receptors and TRPA1, ASIC3 Channels

    Cat # H-130
    Source Synthetic
    MW 311.77
    Target NHE exchangers, TRPA1, ASIC3 channels, P2X7 receptors
    • Bioassay Tested
  • Hongotoxin-1

    A Potent Blocker of Some KV1 K+ Channels

    Cat # STH-400
    MW 4220 Da.
    Target KV1.1, KV1.2, KV1.3 K+ channels
    • Bioassay Tested
  • Huwentoxin-I

    An Antagonist of TTX-Sensitive NaV Channels, N-Type Ca2+ Channels and nAChRs

    Cat # STH-050
    MW 3750 Da.
    Target N-type CaV, TTX-sensitive NaV channels, nAChR
    • Bioassay Tested
  • Huwentoxin-IV

    A Potent Blocker of Neuronal TTX-Sensitive Voltage-Gated NaChannel

    Cat # STH-100
    MW 4106 Da.
    Target TTX-sensitive Na+ channels
    • Bioassay Tested
  • mHuwentoxin-IV

    A Blocker of TTX-Sensitive NaV Channels

    Cat # STH-101
    MW 4089 Da.
    Target TTX-sensitive Na+ channels
    • Bioassay Tested
  • m3-Huwentoxin IV

    A Potent and Selective NaV1.7 Channel Blocker

    Cat # STH-102
    MW 3988 Da.
    Target NaV1.7 channel
    • Bioassay Tested
  • ICA 121431

    A Potent and Selective Blocker of NaV1.3 and NaV1.1 Channels

    Cat # I-170
    Source Synthetic
    MW 449.5
    Target NaV1.1, NaV1.3 channels
    • Bioassay Tested
  • Jingzhaotoxin-V

    A Potent Inhibitor of NaV Channels and KV4.2 and KV4.3 Channels

    Cat # STJ-050
    MW 3605.4 Da.
    Target NaV channels, KV4.2, KV4.3 channels
    • Bioassay Tested
  • Kaliotoxin-1

    A Powerful Blocker of KCa1.1 and certain KV1 Channels

    Cat # STK-370
    MW 4150 Da.
    Target KCa1.1 and some KV1 Kchannels
    • Bioassay Tested
  • KC 12291 hydrochloride

    An Orally Effective Cardioprotective NaV Channel Blocker

    Cat # K-105
    Source Synthetic
    MW 449.99
    Target NaV channels
    • Bioassay Tested
  • Kurtoxin

    A Selective and Potent Blocker of CaV3.1 and CaV3.2 Channels

    Cat # STK-800
    MW 7387 Da.
    Target CaV3.1, CaV3.2 channels
    • Bioassay Tested
  • Kynurenic acid

    An Antagonist of Ionotropic Glutamate Receptors and α7 nAChR

    Cat # K-110
    Source Synthetic
    MW 189.2
    Target iGluR, α7 nAChR
    • Bioassay Tested
  • L-Ascorbic acid

    A Blocker of T-Type CaV Channels

    Cat # L-140
    Source Synthetic
    MW 176.1
    Target T-type Ca2+ channels
    • Bioassay Tested
  • Linopirdine

    A Blocker of KCNQ (KV7) Channels

    Cat # L-155
    Source Synthetic
    MW 391.46
    Target KCNQ K+ channels
    • Bioassay Tested
  • Linopirdine dihydrochloride

    A Blocker of KCNQ (KV7) Channels

    Cat # L-156
    Source Synthetic
    MW 464.39
    Target KCNQ K+ channels
    • Bioassay Tested
  • (-)-Lobeline hydrochloride

    A Potent nAChR Antagonist

    Cat # L-120
    Source Synthetic
    MW 373.9
    Target nAChR
    • Bioassay Tested
  • Mambalgin-1

    A Selective and Reversible ASIC1a Blocker

    Cat # STM-100
    MW 6554.5 Da.
    Target ASIC1 channels
    • Bioassay Tested
  • Mambalgin-2

    A Selective and Reversible ASIC1a Channel Blocker

    Cat # STM-400
    MW 6538 Da.
    Target ASIC1 Channels
    • Bioassay Tested
  • Mambalgin-3

    A Blocker of ASIC1a and ASIC1b Channels

    Cat # STM-500
    MW 6566 Da.
    Target ASIC1a and ASIC1b channels
    • Bioassay Tested
  • MCD peptide

    A Potent and Selective Blocker of KV1.1 and KV1.2 Channels

    Cat # STM-250
    MW 2588 Da.
    Target KV1.1, KV1.2 K+ channels
    • Bioassay Tested
  • Mibefradil dihydrochloride hydrate

    A Blocker of T-type CaV, Orai1-3, and KV10.1 Channels

    Cat # M-150
    Source Synthetic
    MW 568.55
    Target CaV3, Orai1-3, KV10.1 channels
    • Bioassay Tested
  • (+)-MK 801 maleate

    An Antagonist of NMDA Receptors

    Cat # M-230
    Source Synthetic
    MW 337.4
    Target NMDA receptors
    • Bioassay Tested
  • ML 218

    A Selective Blocker of T-type Channels

    Cat # M-165
    Source Synthetic
    MW 369.3
    Target T-type CaV channels
    • Bioassay Tested
  • ML 218 hydrochloride

    A Selective Blocker of T-type Channels

    Cat # M-166
    Source Synthetic
    MW 405.8
    Target T-type CaV channels
    • Bioassay Tested
  • NaV1.7-Compound 36

    A Potent and Selective Blocker of NaV1.7 Channels

    Cat # CMN-003
    Source Synthetic.
    MW 486.85
    Target NaV1.7 channels
    • Bioassay Tested
  • NBQX

    An Antagonist of AMPA/Kainate Receptors

    Cat # N-185
    Source Synthetic
    MW 336.3
    Target AMPA/Kainate receptors
    • Bioassay Tested
  • NBQX disodium salt

    An Antagonist of AMPA/Kainate Receptors

    Cat # N-186
    Source Synthetic
    MW 380.2
    Target AMPA/Kainate receptors
    • Bioassay Tested
  • N-Me-aminopyrimidinone 9

    A Specific Blocker of NaV1.7 Channel

    Cat # N-310
    Source Synthetic
    MW 303.4
    Target NaV1.7 channels
    • Bioassay Tested
  • NNC 55-0396 dihydrochloride

    A Blocker of T-type CaV Channels

    Cat # N-205
    Source Synthetic
    MW 564.57
    Target T-type CaV channels
    • Bioassay Tested
  • NNC 55-0396 dihydrochloride hydrate

    A Blocker of T-type CaV Channels

    Cat # N-206
    Source Synthetic
    MW 573.48
    Target T-type CaV channels
    • Bioassay Tested
  • NS8593

    A Blocker of KCa2 and TRPM7 Channels

    Cat # N-196
    Source Synthetic
    MW 263.3
    Target SK K+ channels, TRPM7
    • Bioassay Tested
  • NS8593 hydrochloride

    A Blocker of KCa2 and TRPM7 Channels

    Cat # N-195
    Source Synthetic
    MW 299.79
    Target SK K+ channels, TRPM7
    • Bioassay Tested
  • Oroxylin A

    An Antagonist of GABA(A) Receptors

    Cat # O-160
    Source Natural
    MW 284.26
    Target GABA(A) receptors
    • Bioassay Tested
  • OsK-1 Toxin

    A Potent Blocker of KV1.3 and KCa3.1 K+ Channels

    Cat # STO-150
    MW 4205 Da.
    Target KV1.1, KV1.2, KV1.3, and KCa3.1 K+ channels
    • Bioassay Tested
  • PD 173212

    A Novel Blocker of N-type CaV Channels

    Cat # P-105
    Source Synthetic
    MW 599.9
    Target N-type Ca2+ channels
    • Bioassay Tested
  • PF-04856264

    A Specific Blocker of NaV1.7 Channel

    Cat # P-265
    Source Synthetic
    MW 437.5
    Target NaV1.7 channels
    • Bioassay Tested
  • PF-05089771

    A Potent and Selective Blocker of NaV1.7 Channel

    Cat # P-315
    Source Synthetic
    MW 500.34
    Target NaV1.7 channels
    • Bioassay Tested
  • PF-05186462

    A Potent and Selective Blocker of NaV1.7 Channels

    Cat # P-365
    Source Synthetic
    MW 531.89
    Target NaV1.7 channels
    • Bioassay Tested
  • PF-05241328

    A Potent and Selective Blocker of NaV1.7 Channels

    Cat # P-345
    Source Synthetic
    MW 436.91
    Target NaV1.7 channels
    • Bioassay Tested
  • Phlo1a

    A Blocker of NaV1.7 Channels

    Cat # STP-350
    MW 4107 Da.
    Target NaV1.7 channels
    • Bioassay Tested
  • Phlo1b

    A Blocker of NaV1.7 Channels

    Cat # STP-370
    MW 4140 Da.
    Target NaV1.7 channels
    • Bioassay Tested
  • Phrixotoxin-1

    A Potent Blocker of KV4.2 and KV4.3 Channels

    Cat # STP-700
    MW 3549 Da.
    Target KV4.2, KV4.3 channels
    • Bioassay Tested
  • Picrotoxin

    An Antagonist of GABA(A), Glycine, and 5-HT3 Receptors

    Cat # P-325
    Source Natural
    MW 602.58
    Target GABA(A), Glycine, 5-HT3 receptors
    • Bioassay Tested
  • Pilsicainide hydrochloride

    A Use-Dependent Anti-Arrhythmic NaV Channel Blocker

    Cat # P-145
    Source Synthetic
    MW 308.85
    Target TTX-Sensitive NaV channels
    • Bioassay Tested
  • PLTX-II

    An Inhibitor of CaV Channels

    Cat # P-510
    MW 5109 Da.
    Target CaV Ca2+ channels
  • ProTx-I

    A Blocker of NaV, CaV3.1, KV2.1 and TRPA1 Channels

    Cat # STP-400
    MW 3988 Da.
    Target NaV, CaV3.1, KV2.1, TRPA1 channels
    • Bioassay Tested
  • ProTx-II

    A Blocker of NaV1.7 and NaV1.5 Channels and Some T-Type Ca2+ Channels

    Cat # STP-100
    MW 3826.6 Da.
    Target NaV channels and T-type Ca2+ channels
    • Bioassay Tested
  • ProTx-II-Biotin

    A Blocker of NaV1.7 and NaV1.5 Channels and some T-Type Ca2+ Channels Conjugated to Biotin

    Cat # STP-100-B
    MW 4053 Da.
    Target NaV Na+ channels and T-type Ca2+ channels
    • Bioassay Tested
  • ProTx-III

    A Potent Blocker of NaV1.7 Channels

    Cat # STP-150
    MW 3802 Da.
    Target NaV1.7 channels
    • Bioassay Tested
  • Psalmotoxin-1

    A Potent Blocker of ASIC1a Channels

    Cat # STP-200
    MW 4689.5 Da.
    Target ASIC1a channels
    • Bioassay Tested
  • Pyrrolopyrimidine 48

    A Blocker of NaV1.7 and NaV1.5 Channel

    Cat # P-275
    Source Synthetic
    MW 385.46
    Target NaV1.7, NaV1.5 channels
    • Bioassay Tested
  • RO-3

    A Potent and Selective Antagonist of P2X3 and P2X2/3 Receptors

    Cat # R-190
    Source Synthetic
    MW 302.37
    Target P2X3 receptors
    • Bioassay Tested
  • Ro 25-6981 maleate

    A Potent and Selective Antagonist of GluN2B-Containing NMDA Receptors

    Cat # R-180
    Source Synthetic
    MW 455.55
    Target GluN2B
    • Bioassay Tested
  • Ro-51

    A Highly Potent and Selective Antagonist of P2X3 and P2X2/3 Receptors

    Cat # R-195
    Source Synthetic
    MW 474.29
    Target P2X3 receptors
    • Bioassay Tested
  • Roscovitine

    A Cyclin-Dependent Kinase (CDK) Inhibitor and a T-Type CaV Channel Blocker

    Cat # R-300
    Source Synthetic
    MW 354.46
    Target CDKs, T-type CaV channels
    • Bioassay Tested
  • SB-366791

    A Specific and Potent TRPV1 Blocker

    Cat # S-180
    Source Synthetic
    MW 287.7
    Target TRPV1 channels
    • Bioassay Tested
  • SB-705498

    A Blocker of TRPV1 Channels

    Cat # S-160
    Source Synthetic
    MW 428.05
    Target TRPV1 channels
    • Bioassay Tested
  • Scyllatoxin

    A Potent Blocker of KCa2 (SK) K+ Channels

    Cat # STS-370
    MW 3423 Da.
    Target KCa2 K+ channels
    • Bioassay Tested
  • sFTX-3.3

    A Blocker of P-Type CaV Channels

    Cat # F-130
    Source Synthetic
    MW 287.4
    Target P-type Ca2+ channels
    • Bioassay Tested
  • SKF 96365 hydrochloride

    A Blocker of CaV3 and TRPC channels and STIM1

    Cat # S-175
    Source Synthetic
    MW 402.9
    Target CaV3 channels, TRPC, STIM1
    • Bioassay Tested
  • SNX-482

    A Blocker of CaV2.3 and KV4.3 Channels

    Cat # RTS-500
    MW 4495 Da.
    Target CaV2.3, CaV2.1, KV4.2, KV4.3 channels
    • Bioassay Tested
  • Spinoxin

    A Potent Blocker of KV1.2 and KV1.3 Channels

    Cat # STS-500
    MW 3701.2 Da.
    Target KV1.2, KV1.3 channels
    • Bioassay Tested
  • ShK (Stichodactyla Toxin)

    A Blocker of KV Channels

    Cat # STS-400
    MW 4055 Da.
    Target Various KV K+ channels
    • Bioassay Tested
  • Stichodactyla Toxin-ATTO Fluor-590

    Fluorescent ShK Conjugate for Sensitive Detection of KV Channels

    Cat # STS-400-AR
    MW ~ 4627 Da.
    Target KV1.1, KV1.3, KV1.4, KV1.6 channels
    • Bioassay Tested
  • Tamapin

    A Blocker of KCa2 Channels

    Cat # STT-400
    MW 3458.16 Da.
    Target KCa2 K+ channels
    • Bioassay Tested
  • TCN 213

    An Antagonist of NMDA Receptors

    Cat # T-215
    Source Synthetic
    MW 376.54
    Target NMDA receptors
    • Bioassay Tested
  • Tertiapin

    A Blocker of Inward Rectifier (Kir) K+ Channels

    Cat # STT-250
    MW 2455 Da.
    Target Kir1.1, Kir3.2 K+ channels
    • Bioassay Tested
  • Tertiapin-LQ

    A Blocker of Kir1.1, Kir3.1 and Kir3.4 K+ Channels 

    Cat # STT-220
    MW 2428 Da.
    Target Kir1.1, Kir3.1, Kir3.4 K+ channels
    • Bioassay Tested
  • Tertiapin-Q

    A Potent Blocker of Inward Rectifier (Kir) K+ Channels

    Cat # STT-170
    MW 2452 Da.
    Target Kir1.1, Kir3.2 Kchannels
    • Bioassay Tested
  • Tertiapin-Q-ATTO Fluor-488

    An Inward Rectifier K+ Channel Blocker Conjugated to the Fluorescent Dye ATTO-488

    Cat # STT-170-AG
    MW 3195.5 Da.
    Target Kir1.1, Kir3.2 Kchannels
    • Bioassay Tested
  • Tertiapin-Q-ATTO Fluor-633

    An Inward Rectifier K+ Channel Blocker Conjugated to the Fluorescent Dye ATTO-633

    Cat # STT-170-FR
    MW 3159.6 Da.
    Target Kir1.1, Kir3.2 Kchannels
    • Bioassay Tested
  • Tracazolate hydrochloride

    A Modulator of GABA(A) Receptors

    Cat # T-230
    Source Synthetic
    MW 340.85
    Target GABA(A) receptors
    • Bioassay Tested
  • TTA-A2

    A Blocker of T-Type CaV Channels

    Cat # T-140
    Source Synthetic
    MW 378.39
    Target T-type CaV channels
    • Bioassay Tested
  • TTA-P2

    A Blocker of T-Type CaV Channels

    Cat # T-155
    Source Synthetic
    MW 431
    Target T-type CaV channels
    • Bioassay Tested
  • TTA-P2 (S-enantiomer)

    A Blocker of T-Type CaV Channels

    Cat # T-210
    Source Synthetic
    MW 431
    Target CaV3 channels
    • Bioassay Tested
  • Waglerin-1

    A Potent Antagonist of nAChR and a Modulator of GABA(A) Receptors

    Cat # STW-001
    MW 2520 Da.
    Target nAChR, GABA(A) receptors
    • Bioassay Tested
  • XE991

    A Blocker of KCNQ Channels

    Cat # X-100
    Source Synthetic
    MW 376.45
    Target KCNQ K+ channels
    • Bioassay Tested
  • XE991 dihydrochloride

    A Blocker of KCNQ Channels

    Cat # X-101
    Source Synthetic
    MW 449.37
    Target KCNQ K+ channels
    • Bioassay Tested
  • XEN907

    A Specific Blocker of NaV1.7 Channels

    Cat # X-105
    Source Synthetic
    MW 351.1
    Target NaV1.7 channels
    • Bioassay Tested
  • CaV Channel Blockers for Pain Research Explorer Kit

    A Screening Package of CaV Channel Blockers for Pain Research Economically Priced

    Cat # EK-385
  • Classical Ion Channel Blockers for Pain Research Explorer Kit

    A Screening Package of Classical Ion Channel Blockers for Pain Research Economically Priced

    Cat # EK-355
  • GABA(A) Receptor Modulator Explorer Kit

    A Screening Package of GABA(A) Receptor Modulators Economically Priced

    Cat # EK-360
  • K+ Channel Blockers for Pain Research Explorer Kit

    A Screening Package of K+ Channel Blockers for Pain Research Economically Priced

    Cat # EK-390
  • KCNQ (KV7) Channel Modulator Explorer Kit

    A Screening Package of KCNQ (KV7) Channel Modulators Economically Priced

    Cat # EK-131
  • KV Channel Blockers for Pain Research Explorer Kit

    A Screening Package of KV Channel Blockers for Pain Research Economically Priced

    Cat # EK-380
  • NaV Channel Blockers for Pain Research Explorer Kit

    A Screening Package of NaV Channel Blockers for Pain Research Economically Priced

    Cat # EK-375
  • NMDA Receptor Antagonist Explorer Kit

    A Screening Package of NMDA Receptor Antagonists Economically Priced

    Cat # EK-350
  • TRPV1 Channel Blocker Explorer Kit

    A Screening Package of TRPV1 Channel Blockers Economically Priced

    Cat # EK-117
  • P2X7 Receptor Basic Research Pack

    All You Need for P2X7 Receptor Research

    Cat # ESB-710
  • P2X7 Receptor Premium Research Pack

    All You Need for P2X7 Receptor Research

    Cat # ESP-710
  • P2X7 Receptor Deluxe Research Pack

    All You Need for P2X7 Receptor Research

    Cat # ESD-710
  • TRPA1 Channel Basic Research Pack

    All You Need for TRPA1 Channel Research

    Cat # ESB-302

* See product page

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