Activators

Voltage-Gated Na+ Channels

Activators

Voltage-gated Na­­­­­­­+ (NaV) channels are important for the generation and propagation of signals in electrically excitable tissues like the muscle, heart, and nerve. Activation of these channels ultimately leads to muscular contraction, cardiac rhythm, and neuronal firing. Nine mammalian isoforms of voltage-gated Na­­­­­­­+ channels have been identified (NaV1.1-NaV1.9). Nine genes (SCN1A, SCN2A, etc.) encoding distinct α subunit isoforms and 4 β subunit genes (SCN1B, SCN2B, etc.) have been identified in the human genome. The nine isoforms share a similar (but complex) architecture.

Displaying 1 to 20 (out of 25 products)
  • 1Kα-Pompilidotoxin

    An Activator of NaV Channels

    Cat # P-172
    Source Synthetic peptide
    MW 1502 Da.
    Target NaV Na+ channels
  • 1Kβ-Pompilidotoxin

    An Activator of NaV Channels

    Cat # P-182
    Source Synthetic peptide
    MW 1531 Da.
    Target NaV Na+ channels
  • 3Rα-Pompilidotoxin

    An Activator of NaV Channels

    Cat # P-174
    Source Synthetic peptide
    MW 1558 Da.
    Target NaV Na+ channels
  • 3R12Rα-Pompilidotoxin

    An Activator of NaV Channels

    Cat # P-176
    Source Synthetic peptide
    MW 1586 Da.
    Target NaV Na+ channels
  • α-Pompilidotoxin

    An Enhancer of NaV Currents

    Cat # P-170
    Source Synthetic peptide
    MW 1529 Da.
    Target TTX-sensitive Nachannels
  • β-Pompilidotoxin

    An Enhancer of NaV Currents

    Cat # P-180
    Source Synthetic peptide
    MW 1559 Da.
    Target TTX-sensitive Na+ channels
  • AaH1 Toxin

    A Potent NaV Channel Inhibitor of Inactivation

    Cat # STA-155
    Source Synthetic peptide.
    MW 6804 Da.
    Target NaV channels
    • New
    • Lyophilized Powder
    • Bioassay Tested
  • Aconitine

    An Activator of NaV Channels

    Cat # A-150
    Source Natural
    MW 645.74
    Target NaV Na+ channels
  • Anthopleurin-C

    A Potent Activator of NaV Channels

    Cat # A-400
    Source Natural peptide
    MW 4884 Da.
    Target NaV channels
  • ATX-II

    A Modulator of NaV Channels

    Cat # STA-700
    Source Synthetic peptide
    MW 4935 Da.
    Target Various NaV channels
  • BDS-I

    A Blocker of KV3 Channels and a Modulator of NaV Channels

    Cat # STB-400
    Source Synthetic peptide
    MW 4708 Da.
    Target KV3.4 K+ channels, NaV Na+ channels
  • BmKI Toxin

    An Activator of NaV Channels

    Cat # STB-100
    Source Synthetic Peptide
    MW 7217 Da.
    Target NaV1.4, NaV1.5, NaV1.6
    • New
    • Lyophilized Powder
    • Bioassay Tested
  • Hm1a

    A Selective and Potent Activator of NaV1.1 Channels

    Cat # STH-601
    Source Synthetic peptide
    MW 3996.4 Da.
    Target NaV1.1 channels
  • Jingzhaotoxin-II

    An Activator of NaV Channels

    Cat # STJ-150
    Source Synthetic peptide
    MW 3561 Da.
    Target NaV Na+ Channels
  • NaV1.1-Compound 3a

    A Modulator of NaV1.1 Channel

    Cat # CMN-002
    Source Synthetic
    MW 344.41
    Target NaV1.1 channels
  • Tf2 Toxin

    A Specific NaV1.3 Channel Opener

    Cat # STT-050
    Source Synthetic peptide
    MW 6954 Da.
    Target NaV1.3 channel
  • Veratridine

    An Enhancer of NaV Channel Activity and an Inducer of Transmitter Release

    Cat # V-110
    Source Natural
    MW 673.8
    Target Various NaV Na+ channels
  • NaV Channel Activator Explorer Kit

    A Screening Package of NaV Channel Activators Economically Priced

    Cat # EK-203
    • Lyophilized Powder
    • Bioassay Tested
    • Shipped at Room Temp.
    • 100% Net Peptide
  • Ion Channel Activators for Pain Research Explorer Kit

    A Screening Package of Ion Channel Activators for Pain Research Economically Priced

    Cat # EK-395
    • Lyophilized Powder
    • Bioassay Tested
    • Shipped at Room Temp.
    • 100% Net Peptide
  • NaV1.2 Channel Basic Research Pack

    All You Need for NaV1.2 Channel Research

    Cat # ESB-002
    • Lyophilized Powder
    • Antigen Incl.
    • Bioassay Tested
    • Shipped at Room Temp.
    • 100% Net Peptide

* See product page

Displaying 1 to 20 (out of 25 products)