Agonists

Adrenergic Receptors

Agonists

Adrenergic Receptors (Adrenoceptors) are seven transmembrane proteins belonging to the superfamily of GPCRs. They respond to the endogenous ligands adrenaline and noradrenaline by inducing a cascade of physiological effects. These receptors have a central role in blood pressure and smooth muscle relaxation and heart contraction. After Rhodopsin, they have become the most studied GPCR to date and are targets for the continuous development of agonists/antagonists.

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  • Amitriptyline hydrochloride

    A Blocker of L-type CaV Channels, an Antagonist of 5-HT2 Serotonin Receptors, and an Agonist of α-Adrenoceptors

    Cat # A-155
    Source Synthetic
    MW 313.86
    Target L-type Ca2+ channels, α-adrenergic receptors, 5-HT2 serotonin receptors

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