Agonists

GABA(A) Receptors

Agonists

GABA(A) Receptors are ionototropic γ-aminobutyric acid type A receptors. Most of the fast inhibitory synaptic transmissions in the brain are mediated by these ligand-gated ion channels in response in to γ-aminobutyric binding.
To date 19 GABA(A) receptors have been cloned in the mammalian central nervous system (CNS) and are classified by their sequence identity into 7 different subunits (α, β, γ, δ, ε, π, and θ). They consist of pentameric structures assembled by different subunits which are mainly permeable to Cl that act to reduce neuronal excitation.

Displaying 1 to 20 (out of 24 products)
  • 2’MeO6MF

    A Potentiator of GABA(A) Receptors

    Cat # M-245
    Source Synthetic
    MW 266.3
    Target GABA(A) receptors
    • New
    • Lyophilized Powder
  • γ-Aminobutyric acid

    A Ligand of GABA(A), GABA(B) Receptors and GABA Transporters

    Cat # G-110
    Source Synthetic
    MW 103.1
    Target GABA(A), GABA(B) receptors, GABA transporters
    • Lyophilized Powder
  • AA 29504

    A Positive Modulator of GABA(A) Receptors

    Cat # A-370
    Source Synthetic
    MW 327.43
    Target GABA(A) receptors
    • Lyophilized Powder
  • CGS 20625

    A Partial Agonist of GABA(A) Receptors

    Cat # C-390
    Source Synthetic
    MW 309.36
    Target GABA(A) receptors
    • Lyophilized Powder
  • Chlormethiazole hydrochloride

    A Positive Modulator of GABA(A) and Glycine Receptors

    Cat # C-360
    Source Synthetic
    MW 198.11
    Target GABA(A), Glycine receptors
    • Lyophilized Powder
  • Diazepam

    An Agonist of GABA(A) Receptors

    Cat # D-215
    Source Synthetic
    MW 284.74
    Target GABA(A) receptors
    • Lyophilized Powder
  • Ganaxolone

    A Selective Positive Modulator of GABA(A) Receptors

    Cat # G-120
    Source Synthetic
    MW 332.5
    Target GABA(A) receptors
    • Lyophilized Powder
  • Isoguvacine hydrochloride

    An Agonist of GABA(A) Receptors

    Cat # I-185
    Source Synthetic
    MW 163.6
    Target GABA(A) receptors
    • Lyophilized Powder
  • Ivermectin

    A Positive Allosteric Modulator of α7 nAChR and of human P2X4 Receptor

    Cat # I-110
    Source Synthetic
    MW 875.09
    Target α7 nAChR, P2X, GABA(A)R
    • Lyophilized Powder
  • Lorazepam

    An Agonist of GABA(A) Receptors

    Cat # L-230
    Source Synthetic
    MW 321.16
    Target GABA(A) receptors
    • Lyophilized Powder
  • MmTx1 Toxin

    A Super Potent Allosteric Modulator of GABA(A) Receptors

    Cat # STM-550
    Source Synthetic peptide
    MW 7205 Da.
    Target GABA(A) receptors
    • Lyophilized Powder
  • MmTx1 Toxin-ATTO-488

    A Super Potent Allosteric Modulator of GABA(A) Receptors Conjugated to the Fluorescent Dye ATTO-488

    Cat # STM-550-AG
    Source Synthetic peptide
    MW ~7775 Da.
    Target GABA(A) receptors
    • New
    • Lyophilized Powder
  • MmTx2 Toxin

    A Super Potent Allosteric Modulator of GABA(A) Receptors

    Cat # STM-600
    Source Synthetic peptide
    MW 7187 Da.
    Target GABA(A) receptors
    • Lyophilized Powder
  • Muscimol

    A Potent Agonist of GABA(A) Receptor and a Partial Agonist of GABA(A) ρ Receptor

    Cat # M-241
    Source Synthetic
    MW 114.1
    Target GABA(A) receptors
    • Lyophilized Powder
  • Muscimol hydrobromide

    A Potent Agonist of GABA(A) Receptor and a Partial Agonist of GABA(A) ρ Receptor

    Cat # M-240
    Source Synthetic
    MW 195.01
    Target GABA(A) receptors
    • Lyophilized Powder
  • SJM-3

    A Positive Allosteric Modulator of GABA(A) Receptors

    Cat # S-215
    Source Synthetic
    MW 354.4
    Target GABA(A) receptors
    • Lyophilized Powder
  • Tracazolate hydrochloride

    A Modulator of GABA(A) Receptors

    Cat # T-230
    Source Synthetic
    MW 340.85
    Target GABA(A) receptors
    • Lyophilized Powder
  • Waglerin-1

    A Potent Antagonist of nAChR and a Modulator of GABA(A) Receptors

    Cat # STW-001
    Source Synthetic peptide
    MW 2520 Da.
    Target nAChR, GABA(A) receptors
    • Lyophilized Powder
  • Zaleplon

    An Agonist of GABA(A) Receptors

    Cat # Z-140
    Source Synthetic
    MW 305.34
    Target GABA(A) receptors
    • Lyophilized Powder
  • Zolpidem

    An Agonist of GABA(A) Receptors

    Cat # Z-100
    Source Synthetic
    MW 307.39
    Target GABA(A) receptors
    • Lyophilized Powder

* See product page

Displaying 1 to 20 (out of 24 products)