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Agonists

GABA(A) Receptors

Agonists

GABA(A) Receptors are ionototropic γ-aminobutyric acid type A receptors. Most of the fast inhibitory synaptic transmissions in the brain are mediated by these ligand-gated ion channels in response in to γ-aminobutyric binding.
To date 19 GABA(A) receptors have been cloned in the mammalian central nervous system (CNS) and are classified by their sequence identity into 7 different subunits (α, β, γ, δ, ε, π, and θ). They consist of pentameric structures assembled by different subunits which are mainly permeable to Cl that act to reduce neuronal excitation.

Displaying 1 to 20 (out of 25 products)
  • 2’MeO6MF

    A Potentiator of GABA(A) Receptors

    Cat # M-245
    Source Synthetic
    MW 266.3
    Target GABA(A) receptors
    • Bioassay Tested
  • γ-Aminobutyric acid

    A Ligand of GABA(A), GABA(B) Receptors and GABA Transporters

    Cat # G-110
    Source Synthetic
    MW 103.1
    Target GABA(A), GABA(B) receptors, GABA transporters
    • Bioassay Tested
  • AA 29504

    A Positive Modulator of GABA(A) Receptors

    Cat # A-370
    Source Synthetic
    MW 327.43
    Target GABA(A) receptors
    • Bioassay Tested
  • CGS 20625

    A Partial Agonist of GABA(A) Receptors

    Cat # C-390
    Source Synthetic
    MW 309.36
    Target GABA(A) receptors
    • Bioassay Tested
  • Chlormethiazole hydrochloride

    A Positive Modulator of GABA(A) and Glycine Receptors

    Cat # C-360
    Source Synthetic
    MW 198.11
    Target GABA(A), Glycine receptors
    • Bioassay Tested
  • Ganaxolone

    A Selective Positive Modulator of GABA(A) Receptors

    Cat # G-120
    Source Synthetic
    MW 332.5
    Target GABA(A) receptors
    • Bioassay Tested
  • Isoguvacine hydrochloride

    An Agonist of GABA(A) Receptors

    Cat # I-185
    Source Synthetic
    MW 163.6
    Target GABA(A) receptors
    • Bioassay Tested
  • MmTx1 Toxin

    A Super Potent Allosteric Modulator of GABA(A) Receptors

    Cat # STM-550
    MW 7205 Da.
    Target GABA(A) receptors
    • Bioassay Tested
  • MmTx1 Toxin-ATTO Fluor-488

    A Super Potent Allosteric Modulator of GABA(A) Receptors Conjugated to the Fluorescent Dye ATTO-488

    Cat # STM-550-AG
    MW ~7775 Da.
    Target GABA(A) receptors
    • Bioassay Tested
  • MmTx2 Toxin

    A Super Potent Allosteric Modulator of GABA(A) Receptors

    Cat # STM-600
    MW 7187 Da.
    Target GABA(A) receptors
    • Bioassay Tested
  • Muscimol

    A Potent Agonist of GABA(A) Receptor and a Partial Agonist of GABA(A) ρ Receptor

    Cat # M-241
    Source Synthetic
    MW 114.1
    Target GABA(A) receptors
    • Bioassay Tested
  • Muscimol hydrobromide

    A Potent Agonist of GABA(A) Receptor and a Partial Agonist of GABA(A) ρ Receptor

    Cat # M-240
    Source Synthetic
    MW 195.01
    Target GABA(A) receptors
    • Bioassay Tested
  • SJM-3

    A Positive Allosteric Modulator of GABA(A) Receptors

    Cat # S-215
    Source Synthetic
    MW 354.4
    Target GABA(A) receptors
    • Bioassay Tested
  • Tracazolate hydrochloride

    A Modulator of GABA(A) Receptors

    Cat # T-230
    Source Synthetic
    MW 340.85
    Target GABA(A) receptors
    • Bioassay Tested
  • Waglerin-1

    A Potent Antagonist of nAChR and a Modulator of GABA(A) Receptors

    Cat # STW-001
    MW 2520 Da.
    Target nAChR, GABA(A) receptors
    • Bioassay Tested

* See product page

Displaying 1 to 20 (out of 25 products)