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5-HT3 Receptors (Serotonin gated channels)

Antagonists

The 5-HT3 receptor is formed by five subunits arranged around a pore forming unit. Receptors could be either monomeric, such as 5-HT3A or heteromeric entities like 5-HT3A/B. Indeed, the type of channel formed displays different pharmacological and electrophysiological characteristics. To date, five 5-HT3 subunits have been identified 5-HT3A-E, which show variability in the N-terminus and in the transmembrane region. 5-HT3A and 5-HT3B are the best characterized among the different types.

Displaying 1 to 22 products (out of 22 products)
  • 3-AQC

    An Antagonist of 5-HT3 Channels

    Cat # A-205
    Source Synthetic
    MW 395.41
    Target 5-HT3A channel
    • Bioassay Tested
  • 5-Hydroxyindole

    A Modulator of 5-HT3 Receptors

    Cat # H-115
    Source Synthetic
    MW 133.15
    Target 5-HT3 receptors
    • Bioassay Tested
  • Azasetron

    A Potent and Selective Antagonist of 5-HT3 Channels

    Cat # A-240
    Source Synthetic
    MW 349.8
    Target 5-HT3A, 5-HT3B
    • Bioassay Tested
  • Azasetron hydrochloride

    A Potent Antagonist of Serotonin-Gated Channels

    Cat # Y-100
    Source Synthetic
    MW 386.3
    Target 5-HT3 receptors
    • Bioassay Tested
  • Bilobalide

    An Antagonist of 5-HT3A and GABA(A) Receptors

    Cat # B-145
    Source Natural
    MW 326.3
    Target 5-HT3A, GABA(A) receptors
    • Bioassay Tested
  • Ginkgolide B

    An Antagonist of 5-HT3A Channels

    Cat # G-170
    Source Natural
    MW 424.4
    Target 5-HT3A receptors
    • Bioassay Tested
  • Lerisetron

    A Potent Antagonist of 5-HT3 Channels

    Cat # L-175
    Source Synthetic
    MW 292.4
    Target 5-HT3A receptors
    • Bioassay Tested
  • LY278584

    A Potent Antagonist of 5-HT3 Receptors

    Cat # L-180
    Source Synthetic
    MW 298.38
    Target 5-HT3 receptors
    • Bioassay Tested
  • MCI-225

    A Potent Antagonist of 5-HT3 Channels and a Selective Noradrenaline Reuptake Inhibitor

    Cat # M-190
    Source Synthetic
    MW 328.4
    Target 5-HT3A receptor, NET transporter
    • Bioassay Tested
  • MDL 72222

    An Antagonist of 5-HT3 Receptors

    Cat # M-155
    Source Synthetic
    MW 314.2
    Target 5-HT3 receptor
    • Bioassay Tested
  • Picrotoxin

    An Antagonist of GABA(A), Glycine, and 5-HT3 Receptors

    Cat # P-325
    Source Natural
    MW 602.58
    Target GABA(A), Glycine, 5-HT3 receptors
    • Bioassay Tested
  • PU02

    A Negative Allosteric Modulator of 5-HT3

    Cat # P-165
    Source Synthetic
    MW 292.4
    Target 5-HT3 receptors
    • Bioassay Tested
  • Ricasetron

    A Potent Antagonist of 5-HT3 Receptors

    Cat # R-150
    Source Synthetic
    MW 313.22
    Target 5-HT3 receptors
    • Bioassay Tested
  • SDZ 205-557 hydrochloride

    An Antagonist of 5-HT3 Channels and 5-HT4 Receptors

    Cat # S-145
    Source Synthetic
    MW 337.2
    Target 5-HT3, 5HT4 receptors
    • Bioassay Tested
  • Talipexole dihydrochloride

    An Antagonist of 5-HT3 Channel, an Agonist of D2 Dopamine Receptor and α2-Adrenoceptor

    Cat # B-140
    Source Synthetic
    MW 282.23
    Target 5-HT3, D2 dopamine, α2-adrenoceptor receptors
    • Bioassay Tested
  • Tropanyl-3,5-dimethylbenzoate

    An Antagonist of 5-HT3 Receptors

    Cat # T-135
    Source Synthetic
    MW 273.4
    Target 5-HT3 receptors
    • Bioassay Tested
  • Tropisetron hydrochloride

    A Potent and Selective Antagonist of 5-Hydroxytryptamine Receptor 3A

    Cat # T-125
    Source Synthetic
    MW 320.76
    Target 5-Hydroxytryptamine Receptor 3A
    • Bioassay Tested
  • U 93631

    An Antagonist of GABA(A) and 5-HT3A Receptors

    Cat # U-120
    Source Synthetic
    MW 299.37
    Target GABA(A), 5-HT3A receptors
    • Bioassay Tested
  • VUF 10166

    A Potent Antagonist of 5-Hydroxytryptamine Receptor 3A and 3B, and an Antagonist of H4 Histamine Receptor

    Cat # V-115
    Source Synthetic
    MW 262.74
    Target 5-Hydroxytryptamine Receptor 3A and 3B
    • Bioassay Tested
  • Zacopride hydrochloride

    A Potent Antagonist of 5-HT3 Receptors and an Agonist of 5-HT4 Receptors

    Cat # Z-110
    Source Synthetic
    MW 346.25
    Target 5-HT3, 5-HT4 receptors
    • Bioassay Tested
  • 5-HT3 Receptor Antagonist Explorer Kit

    A Screening Package of 5-HT3 Receptor Antagonists Economically Priced

    Cat # EK-208
  • 5-HT3 Receptor Modulator Explorer Kit

    A Screening Package of 5-HT3 Receptor Modulators Economically Priced

    Cat # EK-209

* See product page

Displaying 1 to 22 products (out of 22 products)