Antagonists

Adrenergic Receptors

Antagonists

Adrenergic Receptors (Adrenoceptors) are seven transmembrane proteins belonging to the superfamily of GPCRs. They respond to the endogenous ligands adrenaline and noradrenaline by inducing a cascade of physiological effects. These receptors have a central role in blood pressure and smooth muscle relaxation and heart contraction. After Rhodopsin, they have become the most studied GPCR to date and are targets for the continuous development of agonists/antagonists.

Displaying 1 to 3 products (out of 3 products)
  • Carvedilol

    A Blocker of KV1.5 and Kir2.3 Channels and an Antagonist of Adrenoceptors

    Cat # C-180
    Source Synthetic
    MW 406.47
    Target KV1.5, Kir2.3 K+ channels, adrenoceptors
  • Mirtazapine

    An Antagonist of 5-HT2, 5-HT3, Histamine H1 Receptors and α2-Adrenoceptor

    Cat # M-130
    Source Synthetic
    MW 265.4
    Target 5-HT3, 5-HT2, Histamine H1, α2 adrenergic receptors
  • Muscarinic Toxin 3

    An Antagonist of M1 and M4 Muscarinic Receptors and Adrenoceptors

    Cat # M-140
    Source Natural protein
    MW 7379 Da.
    Target M1, M4 muscarinic receptors, adrenoceptors

* See product page

Displaying 1 to 3 products (out of 3 products)