Antagonists

Cannabinoid Receptors

Antagonists

Cannabinoids have been used in Eastern medicine for many years as pain relievers. Δ9-tetrahydrocannabinol (THC), the major psychoactive compound in marijuana and hashish, has been shown to interact with two specific cannabinoid receptors: cannabinoid receptor 1 (CB1 Receptor or CB1R) and cannabinoid receptor 2 (CB2 Receptor or CB2R). The cannabinoid receptors can be distinguished by their amino acid sequences, signaling mechanisms, and tissue distributions. Both receptors belong to the G-protein-coupled receptor (GPCR) superfamily.

Displaying 1 to 2 products (out of 2 products)
  • Cannabichromene

    An Activator of TRPA1 Channels and an Antagonist of Cannabinoid Receptor 1 and TRPM8 Channels

    Cat # C-315
    Source Synthetic
    MW 314.5
    Target TRPA1, TRPM8 channels, Cannabinoid Receptor 1
  • Cannabidiol

    An Activator of TRPV1, TRPV3 and TRPA1 Channels and an Antagonist of Cannabinoid Receptors

    Cat # C-320
    Source Natural
    MW 314.46
    Target TRPV1, TRPV3, TRPA1 channels, CB receptors

* See product page

Displaying 1 to 2 products (out of 2 products)