Antagonists

GPCRs

Antagonists
Displaying 1 to 16 products (out of 16 products)
  • Azilsartan

    An Antagonist of Angiotensin II Receptor Type-1

    Cat # A-245
    Source Synthetic
    MW 456.45
    Target AT1R angiotensin receptors
  • Candesartan

    An Antagonist of Angiotensin II Receptor Type-1 and Angiotensin II Receptor Type-2

    Cat # C-266
    Source Synthetic
    MW 440.45
    Target Angiotensin II receptors
  • Candesartan cilexetil

    An Antagonist of Angiotensin II Receptor Type-1 and Angiotensin II Receptor Type-2

    Cat # C-265
    Source Synthetic
    MW 610.66
    Target Angiotensin II receptors
  • Cannabichromene

    An Activator of TRPA1 Channels and an Antagonist of Cannabinoid Receptor 1 and TRPM8 Channels

    Cat # C-315
    Source Synthetic
    MW 314.5
    Target TRPA1, TRPM8 channels, Cannabinoid Receptor 1
  • Cannabidiol

    An Activator of TRPV1, TRPV3 and TRPA1 Channels and an Antagonist of Cannabinoid Receptors

    Cat # C-320
    Source Natural
    MW 314.46
    Target TRPV1, TRPV3, TRPA1 channels, CB receptors
  • Chlorpromazine hydrochloride

    An Antagonist of nAChRs and an Antagonist of Dopamine Receptors

    Cat # C-165
    Source Synthetic
    MW 355.32
    Target nAChR, Dopamine receptors
  • EMD 66684

    An Antagonist of Angiotensin II Receptor Type-1

    Cat # E-160
    Source Synthetic
    MW 547.05
    Target AT1R receptors
  • Eprosartan mesylate

    An Antagonist of Angiotensin II Receptor Type I

    Cat # E-145
    Source Synthetic
    MW 520.6
    Target AT1R receptors
  • Losartan potassium

    An Antagonist of Angiotensin Receptor Type-1

    Cat # L-185
    Source Synthetic
    MW 461
    Target AT1R receptors
  • Olmesartan

    An Antagonist of Angiotensin II Receptor Type-1

    Cat # O-125
    Source Synthetic
    MW 446.5
    Target AT1R angiotensin receptors
  • PD 123319 ditrifluoroacetate

    A Potent and Selective Antagonist of Angiotensin II Receptor Type-2

    Cat # P-245
    Source Synthetic
    MW 738.66
    Target AT2R receptors
  • Penfluridol

    A T-Type Ca2+ Channel Blocker and D2 Receptor Antagonist

    Cat # P-135
    Source Synthetic
    MW 523.96
    Target T-type Ca2+ channels, D2 receptor
  • Telmisartan

    An Antagonist of Angiotensin Receptor Type-1

    Cat # T-170
    Source Synthetic
    MW 514.6
    Target AT1R receptors
  • Trifluoperazine dihydrochloride

    A Blocker of KV4.3 channel and an Inhibitor of D1 and D2 Dopamine Receptors

    Cat # T-175
    Source Synthetic
    MW 480.4
    Target KV4.3 channels, D1, D2 dopamine receptors
  • Valsartan

    An Antagonist of Angiotensin Receptor Type-1

    Cat # V-120
    Source Synthetic
    MW 435.5
    Target AT1R receptors
  • WRW4

    A Potent Antagonist of FPR2 and FPR3 G-Protein Coupled Receptors

    Cat # GPW-110
    Source Synthetic peptide
    MW 1104.3 Da.

* See product page

Displaying 1 to 16 products (out of 16 products)