Blockers

Inward Rectifier K+ Channels

Blockers

Inwardly rectifying K+ (Kir) channels have diverse physiological functions depending on their type and their location. To date, 15 Kir subunit genes have been identified and classified into seven subfamilies (Kir1 to Kir7). These subfamilies can be categorized into four functional groups: 1) classical Kir channels (Kir2.x), 2) G-protein gated Kir channels (Kir3.x), 3) ATP-sensitive K+ channels (Kir6.x), and 4) K+-transport channels (Kir1.x, Kir4.x, Kir5.x, and Kir7.x).

Displaying 1 to 16 products (out of 16 products)
  • δ-Dendrotoxin

    A Potent and Specific Blocker of KV1.1 Channels and a Less Potent Blocker of Kir1.1 (ROMK1) Channels

    Cat # D-380
    Source Natural peptide
    MW 6568 Da.
    Target KV1.1, KV1.6 and Kir1.1 K+ channels
  • Carvedilol

    A Blocker of KV1.5 and Kir2.3 Channels and an Antagonist of Adrenoceptors

    Cat # C-180
    Source Synthetic
    MW 406.47
    Target KV1.5, Kir2.3 K+ channels, adrenoceptors
  • Gambogic acid

    Kir2.1 Channel Blocker, Apoptosis Inducer, Caspase Activator and Bcl-2 Inhibitor

    Cat # G-250
    Source Synthetic
    MW 628.75
    Target Caspases, Bcl-2, Bax, CD71, Kir2.1
  • Lq2

    A Potent Blocker of Kir1.1 (ROMK1) Channels

    Cat # RTL-550
    Source Recombinant, E. coli
    MW 4353 Da.
    Target Kir1.1 K+ channels
  • Rosiglitazone

    A Blocker of Kir6.1, KV4.3, TRPM3 and an Activator of TRPC5 and PPAR Ligand

    Cat # R-125
    Source Synthetic
    MW 357.43
    Target KV4, Kir6.1, TRPM3, TRPC5 channels
  • Tertiapin

    A Blocker of Inward Rectifier (Kir) K+ Channels

    Cat # STT-250
    Source Synthetic peptide
    MW 2455 Da.
    Target Kir1.1, Kir3.2 K+ channels
  • Tertiapin-LQ

    A Blocker of Kir1.1, Kir3.1 and Kir3.4 K+ Channels 

    Cat # STT-220
    Source Synthetic modified peptide
    MW 2428 Da.
    Target Kir1.1, Kir3.1, Kir3.4 K+ channels
  • Tertiapin-Q

    A Potent Blocker of Inward Rectifier (Kir) K+ Channels

    Cat # STT-170
    Source Synthetic peptide
    MW 2452 Da.
    Target Kir1.1, Kir3.2 Kchannels
  • Tertiapin-Q-ATTO-488

    An Inward Rectifier K+ Channel Blocker Conjugated to the Fluorescent Dye ATTO-488

    Cat # STT-170-AG
    Source Synthetic peptide
    MW 3195.5 Da.
    Target Kir1.1, Kir3.2 Kchannels
  • Tertiapin-Q-ATTO-633

    An Inward Rectifier K+ Channel Blocker Conjugated to the Fluorescent Dye ATTO-633

    Cat # STT-170-FR
    Source Synthetic peptide
    MW 3159.6 Da.
    Target Kir1.1, Kir3.2 Kchannels
  • VU590 dihydrochloride

    A Blocker of Kir1.1 and Kir7.1 K+ Channels

    Cat # V-130
    Source Synthetic
    MW 561.46
    Target Kir1.1, Kir7.1 channels
  • VU591

    A Blocker of Kir1.1 Channel

    Cat # V-125
    Source Synthetic
    MW 368.1
    Target Kir1.1 channel
  • VU591 hydrochloride

    A Blocker of Kir1.1 Channel 

    Cat # V-126
    Source Synthetic
    MW 404.8
    Target Kir1.1 channel
  • Cardiac Channel Blocker Explorer Kit

    A Screening Package of Cardiac Channel Blockers Economically Priced

    Cat # EK-345
    • Lyophilized Powder
    • Bioassay Tested
    • Shipped at Room Temp.
    • 100% Net Peptide
  • K+ Channel Blockers for Pain Research Explorer Kit

    A Screening Package of K+ Channel Blockers for Pain Research Economically Priced

    Cat # EK-390
    • Lyophilized Powder
    • Bioassay Tested
    • Shipped at Room Temp.
    • 100% Net Peptide
  • Kir Channel Blocker Explorer Kit

    A Screening Package of Kir Channel Blockers Economically Priced

    Cat # EK-112
    • Lyophilized Powder
    • Bioassay Tested
    • Shipped at Room Temp.
    • 100% Net Peptide

* See product page

Displaying 1 to 16 products (out of 16 products)