Activators

Mechanosensitive Ion Channels

Activators

Mechanosensitive ion channels (MS channels) represent a diverse population of ion channels. Other membrane-associated proteins with different biophysical properties apart from ion channels, specialized cytoskeletal proteins, cell junction molecules and G-protein-coupled receptors and kinases, among many others are also considered mechanosensitive. MS channels integrate a variety of mechanical stimuli such as shear stress, tension, torsion, and compression and translate them into short-term effects (i.e., changes in ion concentrations and voltage) and long-term effects via changes in gene expression.

Displaying 1 to 15 products (out of 15 products)
  • Cannabichromene

    An Activator of TRPA1 Channels and an Antagonist of Cannabinoid Receptor 1 and TRPM8 Channels

    Cat # C-315
    Source Synthetic
    MW 314.5
    Target TRPA1, TRPM8 channels, Cannabinoid Receptor 1
  • Cannabidiol

    An Activator of TRPV1, TRPV3 and TRPA1 Channels and an Antagonist of Cannabinoid Receptors

    Cat # C-320
    Source Natural
    MW 314.46
    Target TRPV1, TRPV3, TRPA1 channels, CB receptors
  • Capsiate

    A TRPA1 and TRPV1 Channel Activator

    Cat # C-255
    Source Natural
    MW 306.4
    Target TRPA1, TRPV1 channels
  • Curcumin

    An Activator of TRPA1 Channels

    Cat # C-230
    Source Natural
    MW 368.4
    Target TRPA1 channels
  • Etodolac

    A Selective Activator of TRPA1 Channel

    Cat # E-140
    Source Synthetic
    MW 287.3
    Target TRPA1 channel
  • Flupirtine Maleate

    A Potent and Selective Modulator of KCNQ Channels

    Cat # F-150
    Source Synthetic
    MW 420.4
    Target KCNQ K+ channels
  • Glibenclamide

    An Activator of TRPA1 Channel and a Blocker of KATP Channels

    Cat # G-150
    Source Synthetic
    MW 494
    Target TRPA1, KATP channels
  • Ligustilide

    An Activator of TRPA1 Channels

    Cat # L-170
    Source Natural
    MW 190.2
    Target TRPA1 channels
  • alpha/beta MitTx

    An Activator of ASIC1-Containing Channels

    Cat # M-100
    Source Natural protein
    MW 20.8 kDa. (α subunit, 7.1 kDa. and β subunit, 13.7 kDa.)
    Target ASIC1 channels
  • Retigabine

    A Potent and Selective Modulator of KCNQ Channels

    Cat # R-100
    Source Synthetic
    MW 303.3
    Target KCNQ2, KCNQ3, and KCNQ4 K+ channels
  • Retigabine dihydrochloride

    A Potent and Selective Modulator of KCNQ Channels

    Cat # R-101
    Source Synthetic
    MW 376.2
    Target KCNQ2, KCNQ3, KCNQ4 K+ channels
  • Ion Channel Activators for Pain Research Explorer Kit

    A Screening Package of Ion Channel Activators for Pain Research Economically Priced

    Cat # EK-395
    • Lyophilized Powder
    • Bioassay Tested
    • Shipped at Room Temp.
    • 100% Net Peptide
  • TRPA1 Channel Activator Explorer Kit

    A Screening Package of TRPA1 Channel Activators Economically Priced

    Cat # EK-123
    • Lyophilized Powder
    • Bioassay Tested
    • Shipped at Room Temp.
  • TRPA1 Channel Modulator Explorer Kit

    A Screening Package of TRPA1 Channel Modulators Economically Priced

    Cat # EK-120
    • Lyophilized Powder
    • Bioassay Tested
    • Shipped at Room Temp.
    • 100% Net Peptide
  • TRPA1 Channel Basic Research Pack

    All You Need for TRPA1 Channel Research

    Cat # ESB-302
    • Lyophilized Powder
    • Antigen Incl.
    • Bioassay Tested
    • Shipped at Room Temp.

* See product page

Displaying 1 to 15 products (out of 15 products)