Agonists

Endothelin Receptors

Agonists

Endothelin, a 21–amino acid peptide, has potent and sustained vasoconstrictive effects on vascular smooth muscle both in vivo and in vitro and is found in three different isoforms. ET-1 binds and activates two G-protein coupled receptors: ET-A and ET-B. While the former has been attributed to vasoconstriction, the role of ET-B depends mostly on its location; on one hand it could promote vasoconstriction and on the other stimulate nitric oxide (NO) release -a known vasodilator.

Displaying 1 to 7 products (out of 7 products)
  • BQ-3020

    A Selective and Potent Endothelin B Receptor Agonist

    Cat # SPE-200
    Source Synthetic peptide
    MW 2006 Da.
    Target ET-B receptor
    • Lyophilized Powder
  • [Ala1,3,11,15] Endothelin-1

    A Potent Agonist of Endothelin B Receptors 

    Cat # SPE-240
    Source Synthetic peptide
    MW 2368 Da.
    Target ET-B receptor
    • Lyophilized Powder
  • IRL-1620

    A Selective and Potent Endothelin B Receptor Agonist

    Cat # SPE-220
    Source Synthetic peptide
    MW 1820 Da.
    Target ET-B receptor
    • Lyophilized Powder
  • Sarafotoxin S6b

    A Non-Selective and Potent Agonist of Endothelin Receptors

    Cat # SPE-160
    Source Synthetic peptide
    MW 2564 Da.
    Target Endothelin receptors
    • Lyophilized Powder
  • Endothelin Receptor Agonist Explorer Kit

    A Screening Package of Endothelin Receptor Agonists Economically Priced

    Cat # EK-255
    • Lyophilized Powder
  • Endothelin Receptor Pharmacology Explorer Kit

    A Screening Package of Endothelin Receptor Pharmacology Economically Priced

    Cat # EK-257
    • Lyophilized Powder
  • Endothelin Receptor Basic Research Pack

    All You Need for Endothelin Receptors Research

    Cat # ESB-940
    • Lyophilized Powder
    • Antigen Incl.

* See product page

Displaying 1 to 7 products (out of 7 products)