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Antagonists

5-HT3 Receptors (Serotonin gated channels)

Antagonists

The 5-HT3 receptor is formed by five subunits arranged around a pore forming unit. Receptors could be either monomeric, such as 5-HT3A or heteromeric entities like 5-HT3A/B. Indeed, the type of channel formed displays different pharmacological and electrophysiological characteristics. To date, five 5-HT3 subunits have been identified 5-HT3A-E, which show variability in the N-terminus and in the transmembrane region. 5-HT3A and 5-HT3B are the best characterized among the different types.

Displaying 1 to 20 (out of 36 products)
  • 3-AQC

    An Antagonist of 5-HT3 Channels

    Cat # A-205
    Source Synthetic
    MW 395.41
    Target 5-HT3A channel
    • Bioassay Tested
  • 5-Hydroxyindole

    A Modulator of 5-HT3 Receptors

    Cat # H-115
    Source Synthetic
    MW 133.15
    Target 5-HT3 receptors
    • Bioassay Tested
  • Azasetron

    A Potent and Selective Antagonist of 5-HT3 Channels

    Cat # A-240
    Source Synthetic
    MW 349.8
    Target 5-HT3A, 5-HT3B
    • Bioassay Tested
  • Azasetron hydrochloride

    A Potent Antagonist of Serotonin-Gated Channels

    Cat # Y-100
    Source Synthetic
    MW 386.3
    Target 5-HT3 receptors
    • Bioassay Tested
  • Bilobalide

    An Antagonist of 5-HT3A and GABA(A) Receptors

    Cat # B-145
    Source Natural
    MW 326.3
    Target 5-HT3A, GABA(A) receptors
    • Bioassay Tested
  • Ginkgolide B

    An Antagonist of 5-HT3A Channels

    Cat # G-170
    Source Natural
    MW 424.4
    Target 5-HT3A receptors
    • Bioassay Tested
  • Lerisetron

    A Potent Antagonist of 5-HT3 Channels

    Cat # L-175
    Source Synthetic
    MW 292.4
    Target 5-HT3A receptors
    • Bioassay Tested
  • LY278584

    A Potent Antagonist of 5-HT3 Receptors

    Cat # L-180
    Source Synthetic
    MW 298.38
    Target 5-HT3 receptors
    • Bioassay Tested
  • MCI-225

    A Potent Antagonist of 5-HT3 Channels and a Selective Noradrenaline Reuptake Inhibitor

    Cat # M-190
    Source Synthetic
    MW 328.4
    Target 5-HT3A receptor, NET transporter
    • Bioassay Tested
  • MDL 72222

    An Antagonist of 5-HT3 Receptors

    Cat # M-155
    Source Synthetic
    MW 314.2
    Target 5-HT3 receptor
    • Bioassay Tested

* See product page

Displaying 1 to 20 (out of 36 products)