Antagonists

Muscarinic Receptors

Antagonists

The action of the neurotransmitter acetylcholine is mediated through two types of receptors, the ionotrophic nicotinic receptors and the metabotrophic muscarinic receptors. The muscarinic receptors belong to the superfamily of 7-TM G-protein-coupled receptors. Five subtypes of muscarinic receptors have been cloned and named m1-m5.
The muscarinic receptors are widely distributed throughout the body, but are predominantly expressed within the parasympathetic nervous system and exerts both excitatory and inhibitory control over central and peripheral tissues.

Displaying 1 to 7 products (out of 7 products)
  • Biperiden hydrochloride

    A Selective Antagonist of M1 Muscarinic Acetylcholine Receptors

    Cat # B-115
    Source Synthetic
    MW 347.92
    Target M1-M5 muscarinic receptors
  • Muscarinic Toxin 3

    An Antagonist of M1 and M4 Muscarinic Receptors and Adrenoceptors

    Cat # M-140
    Source Natural protein
    MW 7379 Da.
    Target M1, M4 muscarinic receptors, adrenoceptors
  • Muscarinic Toxin 7

    An Antagonist of M1 Muscarinic Receptor

    Cat # M-200
    Source Natural protein
    MW 7472 Da.
    Target M1 muscarinic receptor
  • Orphenadrine citrate salt

    An Antagonist of Muscarinic and NMDA Receptors and Voltage-Gated Na+ Channels

    Cat # O-100
    Source Synthetic
    MW 461.5
    Target Muscarinic, H1 histamine, NMDA receptors, NaV Na+ channels
  • Orphenadrine hydrochloride

    An Antagonist of Muscarinic and NMDA Receptors and Voltage-Gated Na+ Channels

    Cat # O-101
    Source Synthetic
    MW 305.8
    Target Muscarinic, H1 histamine, NMDA receptors, NaV Na+ channels
  • Tropicamide

    A Potent Muscarinic Receptor Antagonist

    Cat # T-120
    Source Synthetic
    MW 284.3
    Target M1-M5 muscarinic receptors
  • Muscarinic Receptor Antagonist Explorer Kit

    A Screening Package of Muscarinic Receptor Antagonists Economically Priced

    Cat # EK-206
    • Lyophilized Powder
    • Bioassay Tested
    • Shipped at Room Temp.

* See product page

Displaying 1 to 7 products (out of 7 products)