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Antagonists

NMDA Receptors

Antagonists

The NMDA receptors are members of the glutamate receptor family of ion channels that also include the AMPA and Kainate receptors.
The NMDA receptors are encoded by seven genes: one NMDAR1 (or NR1) subunit, four NR2 (NR2A-NR2D) and two NR3 (NR3A-NR3B) subunits. The functional NMDA receptor appears to be a heterotetramer composed of two NMDAR1 and two NMDAR2 subunits. Whereas the NMDAR2 subunits that assemble with the NMDAR1 subunit can be either of the same kind (i.e. two NMDAR2A subunits) or different (one NMDAR2A with one NMDAR2B). NMDAR3 subunits can substitute the NMDAR2 subunits in their complex with the NMDAR1 subunit.

Displaying 1 to 20 (out of 40 products)
  • 5,7-Dichlorokynurenic acid

    An Antagonist of NMDA Receptors

    Cat # D-190
    Source Synthetic
    MW 258.06
    Target NMDA receptors
    • Bioassay Tested
  • 5,7-Dichlorokynurenic acid monohydrate

    An Antagonist of NMDA Receptors

    Cat # D-191
    Source Synthetic
    MW 276.07
    Target NMDA receptors
    • Bioassay Tested
  • 7-Chlorokynurenic acid

    An Antagonist of NMDA Receptors

    Cat # C-285
    Source Synthetic
    MW 223.61
    Target NMDA receptors
    • Bioassay Tested
  • 7-Chlorokynurenic acid sodium salt

    An Antagonist of NMDA Receptors

    Cat # C-286
    Source Synthetic
    MW 245.59
    Target NMDA receptors
    • Bioassay Tested
  • α-Asarone

    An Antagonist of NaV Channels, GABA(A) Receptors, NMDA Receptors and an Inhibitor of TrkB Receptor

    Cat # A-260
    Source Natural
    MW 208.3
    Target NaV channels, GABA(A) receptors, TrkB receptors, NMDA receptors
    • Bioassay Tested
  • Arcaine sulfate

    An Antagonist of NMDA Receptors

    Cat # A-285
    Source Synthetic
    MW 270.31
    Target NMDA receptors
    • Bioassay Tested
  • CGP-37849

    A Potent and Selective Antagonist of NMDA Receptors

    Cat # C-325
    Source Synthetic
    MW 209.14
    Target NMDA receptors
    • Bioassay Tested
  • CGS 19755

    An NMDA Receptor Antagonist

    Cat # C-310
    Source Synthetic
    MW 223.16
    Target NMDA receptors
    • Bioassay Tested
  • Clobenpropit dihydrobromide

    A Potent and Selective Antagonist of Histamine H3 Receptors and an Antagonist of NMDA Receptors

    Cat # C-345
    Source Synthetic
    MW 470.65
    Target Histamine H3, Histamine H4, NMDA receptors
    • Bioassay Tested
  • CNS-1102

    A Potent NMDA Receptor Antagonist

    Cat # C-305
    Source Synthetic
    MW 339.86
    Target NMDA receptors
    • Bioassay Tested
  • Conantokin G

    A Selective and Competitive Antagonist of GluN2B Receptor

    Cat # STC-666
    MW 2264.2 Da.
    Target GluN2B receptor
    • Bioassay Tested
  • Conantokin R

    An Antagonist of GluN2A and GluN2B Receptors

    Cat # STC-777
    Source Synthetic peptide
    MW 3098 Da.
    Target GluN2B receptor
    • Bioassay Tested
  • (±)-CPP

    An NMDA Receptor Antagonist

    Cat # C-175
    Source Synthetic
    MW 252.2
    Target NMDA receptors
    • Bioassay Tested
  • D-AP5

    A Competitive NMDA Receptor Antagonist

    Cat # D-145
    Source Synthetic
    MW 197.1
    Target NMDA receptors
    • Bioassay Tested
  • DL-AP5

    A Competitive NMDA Receptor Antagonist

    Cat # D-140
    Source Synthetic
    MW 197.1
    Target NMDA receptors
    • Bioassay Tested
  • DL-AP7

    An Antagonist of NMDA Receptors

    Cat # D-200
    Source Synthetic
    MW 225.19
    Target NMDA receptors
    • Bioassay Tested
  • DQP-1105

    A Potent Noncompetitive Antagonist of GluN2D/C-Containing NMDA Receptors

    Cat # D-210
    Source Synthetic
    MW 558.43
    Target GluN2D and GluN2C-containing NMDA receptors
    • Bioassay Tested
  • Eliprodil

    An Antagonist of NMDA Receptors and N- and P-Type CaV Channels

    Cat # E-155
    Source Synthetic
    MW 347.9
    Target NMDA receptors, N-, P-type CaV channels
    • Bioassay Tested
  • Kynurenic acid

    An Antagonist of Ionotropic Glutamate Receptors and α7 nAChR

    Cat # K-110
    Source Synthetic
    MW 189.2
    Target iGluR, α7 nAChR
    • Bioassay Tested

* See product page

Displaying 1 to 20 (out of 40 products)