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CaV2 Channel Blocker Explorer Kit

A Screening Package of CaV2 Channel Blockers Economically Priced
  • Lyophilized Powder
  • Bioassay Tested
Cat #: EK-110
Sizes: 21 Vials
Last update: 24/04/2019

Alomone Labs is pleased to offer the CaV2 Channel Blocker Explorer Kit (#EK-110). The Explorer Kit contains many classical CaV2 channel blockers, ideal for screening purposes.

For research purposes only, not for human use
Compounds
Product Name Cat # Size
α-Conotoxin PeIA
 		STC-970 1 x 0.1 mg
ω-Agatoxin IVA
 		STA-500 1 x 50 µg
ω-Agatoxin TK
 		STA-530 1 x 50 µg
ω-Conotoxin CnVIIA
 		STC-800 1 x 0.1 mg
ω-Conotoxin CVIA
 		STC-750 1 x 50 µg
ω-Conotoxin CVIB
 		STC-410 1 x 50 µg
ω-Conotoxin CVIC
 		STC-420 1 x 50 µg
ω-Conotoxin CVIE
 		STC-760 1 x 50 µg
ω-Conotoxin GVIA
 		C-300 1 x 0.1 mg
ω-Conotoxin MVIIA
 		C-670 1 x 50 µg
ω-Conotoxin MVIIC
 		C-150 1 x 30 µg
ω-Conotoxin MVIID
 		STC-751 1 x 50 µg
ω-Conotoxin RVIA
 		STC-850 1 x 0.1 mg
ω-Conotoxin SO3
 		STC-470 1 x 50 µg
ω-Grammotoxin SIA
 		G-450 1 x 5 µg
Cilnidipine
 		C-135 1 x 5 mg
FTX-3.3
 		F-120 1 x 1 mg
sFTX-3.3
 		F-130 1 x 1 mg
Huwentoxin-I
 		STH-050 1 x 50 µg
PD 173212
 		P-105 1 x 5 mg
SNX-482
 		RTS-500 1 x 25 µg
References
Scientific Background

Voltage-dependent Ca2+ channels (CaV) form an important route for Ca2+ entry into cells upon deviations from the cell's resting membrane potential.  There are ten CaV α1 subunit genes, divided into three subfamilies on both a functional and sequence homology basis. The CaV1 subfamily includes four genes which encode the L-type channels, the CaV3 subfamily includes three genes encoding the T-type channels and the CaV2 subfamily consists of three isoforms encoding P/Q- , N- and R-type channels, with all three contributing to neurotransmitter release in neurons.
References
  1. Catterall, W.A. et al. (2003) Pharmacol. Rev. 55, 579.
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